SCHEMBL7463531

SCHEMBL7463531

[CH2]CCCc1oc(-n2ccnc2C)nc1-c1ccc(Cl)cc1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPKAPK2 P49137 4/20 0.34
GRM5 P41594 1/20 0.32
MAPT P10636 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
GLA P06280 1/20 0.31
GAA P10253 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP19A1 P11511 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
POLB P06746 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
PSEN1 P49768 1/20 0.31
PSEN2 P49810 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL963990 0.89 SIRT2 (0.40) MAPKAPK2KDM4EALDH1A1GLAGAA
SCHEMBL965656 0.88 SIRT2 (0.37) MAPKAPK2KDM4EALDH1A1GLAGAA
SCHEMBL964061 0.87 SIRT2 (0.36) MAPKAPK2CYP3A4CYP2D6KCNH2
SCHEMBL1360344 0.87 SIRT2 (0.36) MAPKAPK2CYP3A4CYP2D6KCNH2
SCHEMBL7460783 0.86 MAPKAPK2 (0.35) MAPKAPK2KDM4EALDH1A1GLAGAA
SCHEMBL7461461 0.85 RXRA (0.43)
SCHEMBL1361100 0.85 PSEN1 (0.33) MAPKAPK2CYP1A2CYP3A4CYP2D6CYP19A1
SCHEMBL7452859 0.84 PSEN1 (0.34) MAPKAPK2ALDH1A1SMN1; SMN2CYP3A4CYP2D6
SCHEMBL1360093 0.84 CYP1A2 (0.42) GRM5MAPTSMN1; SMN2CYP1A2CYP3A4
SCHEMBL1362394 0.84 TDP1 (0.47) MAPTALDH1A1RAB9ASMN1; SMN2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6498179-B1 SUCH AS 4-(4-CHLOROPHENYL)-5-(3-(2-METHOXYPHENOXY)PROPYL)-2-(2-METHYL-1 -IMIDAZOLYL)OXAZOLE; INSULIN SECERTION PROMOTING AND BLOOD SUGAR DEPRESSING EFFECT; DIABETES; LOW TOXICITY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2002-12-24 US disclosed
EP-0891340-B1 OXAZOLE DERIVATIVES, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-11-13 EP disclosed