SCHEMBL7464157

SCHEMBL7464157

CC1(C)CCC(C)(C)c2cc(C(F)(F)F)c(-c3c(Cl)cccc3/C=C3/SC(=O)NC3=O)cc21

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PIM2 Q9P1W9 7/20 0.48
PIM1 P11309 6/20 0.48
PIM3 Q86V86 2/20 0.43
TTR P02766 3/20 0.43
CISD1 Q9NZ45 1/20 0.43
IGF1R P08069 2/20 0.42
PTPN1 P18031 2/20 0.42
ESRRA P11474 3/20 0.41
CYP3A4 P08684 1/20 0.41
NR1H4 Q96RI1 1/20 0.41
HPGD P15428 1/20 0.41
MYC P01106 1/20 0.40
MAX P61244 1/20 0.40
MEN1 O00255 1/20 0.40
AKR1B1 P15121 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7464163 1.00 PIM2 (0.48) PIM2PIM1PIM3TTRCISD1
SCHEMBL7459431 0.89 TTR (0.50) PIM2PIM1TTRCISD1IGF1R
SCHEMBL7459436 0.89 TTR (0.50) PIM2PIM1TTRCISD1IGF1R
SCHEMBL7468506 0.88 PIM1 (0.49) PIM2PIM1TTRCISD1IGF1R
SCHEMBL7468503 0.88 PIM1 (0.49) PIM2PIM1TTRCISD1IGF1R
SCHEMBL7469698 0.87 GSK3B (0.53) PIM2PIM1TTRCISD1IGF1R
SCHEMBL7463047 0.87 ESRRA (0.53) PIM2PIM1PIM3PTPN1ESRRA
SCHEMBL7463041 0.87 ESRRA (0.53) PIM2PIM1PIM3PTPN1ESRRA
SCHEMBL7469695 0.87 GSK3B (0.53) PIM2PIM1TTRCISD1IGF1R
SCHEMBL7465115 0.86 TTR (0.50) PIM2PIM1PIM3TTRIGF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214305-A1 BENZYLIDENE-THIAZOLIDINEDIONES AND ANALOGUES AND THEIR USE IN THE TREATMENT OF INFLAMMATION Maxia Pharmaceuticals, Inc. (US) 2002-06-19 EP claimed
WO-2001016123-A1 BENZYLIDENE-THIAZOLIDINEDIONES AND ANALOGUES AND THEIR USE IN THE TREATMENT OF INFLAMMATION MAXIA PHARMACEUTICALS, INC. (US) 2001-03-08 WO claimed
EP-1214305-A1 BENZYLIDENE-THIAZOLIDINEDIONES AND ANALOGUES AND THEIR USE IN THE TREATMENT OF INFLAMMATION Maxia Pharmaceuticals, Inc. (US) 2002-06-19 EP disclosed
WO-2001016123-A1 BENZYLIDENE-THIAZOLIDINEDIONES AND ANALOGUES AND THEIR USE IN THE TREATMENT OF INFLAMMATION MAXIA PHARMACEUTICALS, INC. (US) 2001-03-08 WO disclosed