SCHEMBL7464625

SCHEMBL7464625

Cc1ccc(CNc2nccc(-c3ccncc3)n2)cc1C

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 11/20 0.52
CLK4 Q9HAZ1 11/20 0.52
CLK1 P49759 8/20 0.52
DYRK1B Q9Y463 8/20 0.52
CLK2 P49760 7/20 0.52
ROCK2 O75116 1/20 0.48
CHEK2 O96017 1/20 0.48
PRKACA P17612 1/20 0.48
RPS6KB1 P23443 1/20 0.48
AKT1 P31749 1/20 0.48
MATK P42679 1/20 0.48
GSK3A P49840 1/20 0.48
GSK3B P49841 1/20 0.48
RPS6KA3 P51812 1/20 0.48
NEK4 P51957 1/20 0.48
ROCK1 Q13464 1/20 0.48
PRKG1 Q13976 1/20 0.48
PKN2 Q16513 1/20 0.48
CDC42BPA Q5VT25 1/20 0.48
HIPK4 Q8NE63 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7467627 0.78 ABL1 (0.61) DYRK1ACLK4CLK1DYRK1BCLK2
SCHEMBL4154191 0.74 IKBKB (0.55)
SCHEMBL4906864 0.73 MKNK1 (0.71) MKNK1HIF1AMKNK2
SCHEMBL7466961 0.71 SRC (0.63) ABL1BCRSRC
SCHEMBL10917879 0.71 ABL1 (0.51) DYRK1AROCK1AURKBABL1BCR
SCHEMBL7471338 0.71 MKNK1 (0.51) DYRK1BROCK2ROCK1PKN2MKNK1
SCHEMBL3654446 0.70 DYRK1A (0.52) DYRK1ACLK4CLK1DYRK1BCLK2
SCHEMBL30299573 0.70 DYRK1A (0.55) DYRK1ACLK4CLK1DYRK1BCLK2
SCHEMBL7465536 0.69 ABL1 (0.54) ABL1BCRSRC
SCHEMBL2580846 0.69 ABL1 (0.74) PRKACAABL1BCRSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0233461-B2 4,5,6-Substituted-2-pyrimidinamines AMERICAN CYANAMID CO (US) 2002-05-29 EP disclosed