SCHEMBL7464802

SCHEMBL7464802

O=C(N1CCc2c(ccc3ccccc23)C1)C(F)(F)F

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 5/20 0.52
ESR2 Q92731 5/20 0.52
KDM4E B2RXH2 1/20 0.42
TAAR1 Q96RJ0 1/20 0.42
ABHD6 Q9BV23 5/20 0.42
PKM P14618 1/20 0.41
RIPK1 Q13546 2/20 0.39
TMPRSS2 O15393 1/20 0.38
HPGD P15428 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7789910 0.87 ESR1 (0.43) ESR1ESR2KDM4ETAAR1ABHD6
Hydrochloric Acid SCHEMBL8384089 0.82 KDM4E (0.45) KDM4ETAAR1TMPRSS2HPGD
SCHEMBL566389 0.76 ESR1 (0.68) ESR1ESR2TAAR1ABHD6RIPK1
SCHEMBL30263783 0.76 ESR1 (0.68) ESR1ESR2TAAR1ABHD6RIPK1
SCHEMBL23553488 0.76 ESR1 (0.52) ESR1ESR2ABHD6
SCHEMBL7637893 0.76 ESR1 (0.56) ESR1ESR2ABHD6PKM
SCHEMBL8177222 0.76 ESR1 (0.56) ESR1ESR2ABHD6PKMRIPK1
SCHEMBL30814383 0.76 ESR1 (0.52) ESR1ESR2ABHD6
SCHEMBL7462013 0.75 ESR1 (0.46) ESR1ESR2ABHD6PKMRIPK1
SCHEMBL7641094 0.75 ABHD6 (0.52) ESR1ESR2ABHD6PKMRIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1003747-A4 CARBAPENEMS WITH NAPHTHOSULTAM DERIVATIVE LINKED VIA METHYLENE MERCK & CO INC (US) 2002-11-06 EP disclosed
EP-1133477-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2001-09-19 EP disclosed
US-6251890-B1 TREATING OR PREVENTING BACTERIAL INFECTIONS IN MAMMALIAN PATIENTS MERCK & CO., INC. 2001-06-26 US disclosed
WO-2000032579-A1 SUBSTITUTED BENZIMIDAZOLES AND THEIR USE AS PARP INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2000-06-08 WO disclosed
EP-1003747-A1 CARBAPENEMS WITH NAPHTHOSULTAM DERIVATIVE LINKED VIA METHYLENE Merck & Co., Inc. (US) 2000-05-31 EP disclosed
WO-1999009032-A1 CARBAPENEMS WITH NAPHTHOSULTAM DERIVATIVE LINKED VIA METHYLENE MERCK & CO., INC. (US) 1999-02-25 WO disclosed