SCHEMBL7789910

SCHEMBL7789910

O=C(N1Cc2ccc3ccccc3c2C1)C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 4/20 0.43
ESR2 Q92731 4/20 0.43
ABHD6 Q9BV23 5/20 0.39
KDM4E B2RXH2 2/20 0.36
TAAR1 Q96RJ0 1/20 0.36
PIK3CA P42336 1/20 0.35
ANPEP P15144 1/20 0.35
HSP90AA1 P07900 1/20 0.35
HSP90AB1 P08238 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GLA P06280 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
RCE1 Q9Y256 1/20 0.35
DPP8 Q6V1X1 2/20 0.34
DPP9 Q86TI2 2/20 0.34
DPP7 Q9UHL4 2/20 0.34
DPP4 P27487 1/20 0.34
NOTUM Q6P988 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7464802 0.87 ESR1 (0.52) ESR1ESR2ABHD6KDM4ETAAR1
SCHEMBL7786861 0.78 ESR1 (0.53) ESR1ESR2ABHD6PIK3CAHSP90AA1
SCHEMBL1367873 0.77 NOTUM (0.55) ESR1ESR2ABHD6TAAR1HSP90AA1
SCHEMBL31277017 0.77 NOTUM (0.55) ESR1ESR2ABHD6TAAR1HSP90AA1
SCHEMBL7529328 0.74 CYP3A4 (0.46) ESR1ESR2ABHD6GAA
SCHEMBL7518323 0.74 ESR1 (0.36) ESR1ESR2ABHD6PIK3CAHSP90AA1
SCHEMBL25825897 0.74 ABHD6 (0.47) ESR1ESR2ABHD6HSP90AA1HSP90AB1
SCHEMBL7524427 0.73 ESR1 (0.44) ESR1ESR2ABHD6NOTUM
SCHEMBL7521814 0.73 HPGD (0.38) ESR1ESR2ALDH1A1GAAMAPT
SCHEMBL7789796 0.73 ESR1 (0.38) ESR1ESR2ABHD6HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6251890-B1 TREATING OR PREVENTING BACTERIAL INFECTIONS IN MAMMALIAN PATIENTS MERCK & CO., INC. 2001-06-26 US disclosed