SCHEMBL7465223

SCHEMBL7465223

Cn1cc(NC(=O)[C@H](CCCNC(=N)N)NC(=O)OC(C)(C)C)cc1-c1nc2cc(C(=O)Nc3ccc(N(CCCl)CCCl)cc3)ccc2[nH]1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRAS P01112 12/20 0.44
ESR1 P03372 12/20 0.44
ESR2 Q92731 12/20 0.44
HDAC4 P56524 2/20 0.35
HDAC1 Q13547 2/20 0.35
HDAC3 O15379 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC11 Q96DB2 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
HDAC9 Q9UKV0 1/20 0.34
HDAC5 Q9UQL6 1/20 0.34
BRD4 O60885 2/20 0.33
SIRT5 Q9NXA8 1/20 0.33
EGFR P00533 1/20 0.33
ERBB2 P04626 1/20 0.33
MLLT1 Q03111 1/20 0.33
ITGB3 P05106 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7467778 0.88 HRAS (0.49) HRASESR1ESR2EGFRERBB2
SCHEMBL7467474 0.83 HRAS (0.47) HRASESR1ESR2BRD4EGFR
Hydrochloric Acid SCHEMBL7465253 0.81 HRAS (0.52) HRASESR1ESR2EGFRERBB2
SCHEMBL7472023 0.80 HRAS (0.51) HRASESR1ESR2EGFRERBB2
Hydrochloric Acid SCHEMBL7475008 0.78 HRAS (0.64) HRASESR1ESR2EGFRERBB2
Hydrochloric Acid SCHEMBL7471999 0.77 HRAS (0.52) HRASESR1ESR2EGFRERBB2
Hydrochloric Acid SCHEMBL7465588 0.77 HRAS (0.46) HRASESR1ESR2EGFR
Hydrochloric Acid SCHEMBL7466261 0.76 HRAS (0.49) HRASESR1ESR2EGFRERBB2
SCHEMBL7467693 0.76 HRAS (0.47) HRASESR1ESR2HDAC1HDAC2
Hydrochloric Acid SCHEMBL7465502 0.75 HRAS (0.58) HRASESR1ESR2EGFRERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0711768-B1 BENZIMIDAZOLE DERIVATIVE MITSUI CHEMICALS INC (JP) 2002-02-13 EP disclosed