SCHEMBL7465273

SCHEMBL7465273

CCCn1cnc2c1c(=O)n(CCCP(=O)(OCC)OCC)c(=O)n2C

nearest known ligand 0.62

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 8/20 0.62
LMNA P02545 1/20 0.62
ESR1 P03372 1/20 0.62
CYP1A2 P05177 1/20 0.62
MAPT P10636 1/20 0.62
NFKB1 P19838 1/20 0.62
ACHE P22303 1/20 0.62
BLM P54132 1/20 0.62
PMP22 Q01453 1/20 0.62
PDE4B Q07343 7/20 0.55
PDE4C Q08493 7/20 0.55
PDE4D Q08499 7/20 0.55
ADORA2A P29274 6/20 0.55
ADORA2B P29275 5/20 0.55
TNF P01375 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7457088 0.97 PDE4A (0.64) PDE4ALMNAESR1CYP1A2MAPT
SCHEMBL7455860 0.96 PDE4A (0.63) PDE4ALMNAESR1CYP1A2MAPT
SCHEMBL7459717 0.92 PDE4A (0.52) PDE4ALMNAESR1CYP1A2MAPT
SCHEMBL7463585 0.92 PDE4A (0.57) PDE4ALMNAESR1CYP1A2MAPT
SCHEMBL7458605 0.91 ADORA2B (0.58) PDE4ALMNAESR1CYP1A2MAPT
SCHEMBL7465863 0.90 PDE4A (0.56) PDE4ALMNAESR1CYP1A2MAPT
SCHEMBL7453497 0.89 PDE4A (0.49) PDE4ALMNAESR1CYP1A2MAPT
SCHEMBL7460890 0.88 ADORA2A (0.60) PDE4ACYP1A2BLMPMP22PDE4B
SCHEMBL8656385 0.88 PDE4A (0.59) PDE4ALMNAESR1CYP1A2MAPT
SCHEMBL7557802 0.88 ADORA2B (0.57) PDE4ALMNAESR1CYP1A2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0771813-B1 Alkylxanthine phosphonates and alkylxanthine phosphine oxydes and their use as medicines HOECHST AG (DE) 2002-01-16 EP disclosed
EP-0771813-A1 Alkylxanthine phosphonates and alkylxanthine phosphine oxydes and their use as medicines HOECHST AKTIENGESELLSCHAFT (DE) 1997-05-07 EP disclosed