SCHEMBL7465368

SCHEMBL7465368

CS(=O)(=O)OCc1cc(Cl)cc([N+](=O)[O-])c1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 8/20 0.41
S1PR4 O95977 1/20 0.38
ALDH1A1 P00352 4/20 0.38
TDP1 Q9NUW8 1/20 0.38
POLB P06746 2/20 0.37
HTT P42858 1/20 0.37
TSHR P16473 2/20 0.35
MAPT P10636 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
MEN1 O00255 1/20 0.34
LMNA P02545 1/20 0.34
KMT2A Q03164 1/20 0.34
TXNRD1 Q16881 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18407634 0.85 TSHR (0.45) CYP19A1ALDH1A1POLBHTTTSHR
SCHEMBL7019884 0.84 POLB (0.39) CYP19A1ALDH1A1POLBHTTTSHR
SCHEMBL7013539 0.83 TSHR (0.52) CYP19A1POLBHTTTSHRMAPT
SCHEMBL4426073 0.82 IDO1 (0.48) ALDH1A1TSHRMAPTLMNA
SCHEMBL13722513 0.80 HTT (0.43) CYP19A1S1PR4ALDH1A1TDP1POLB
SCHEMBL787701 0.78 GAA (0.38) ALDH1A1TDP1POLBTSHRMAPT
SCHEMBL5005099 0.77 POLB (0.52) ALDH1A1POLBHTTMAPTSMN1; SMN2
SCHEMBL20511401 0.77 TSHR (0.54) CYP19A1ALDH1A1POLBHTTTSHR
SCHEMBL3087323 0.76 FFAR4 (0.43) MEN1KMT2A
SCHEMBL28743760 0.76 HTT (0.41) ALDH1A1HTTMAPTSMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0930298-B1 FLUORINATED 1,4-DISUBSTITUTED PIPERIDINE DERIVATIVES BANYU PHARMA CO LTD (JP) 2002-12-18 EP disclosed
US-6040449-A USEFUL FOR FORMING FLUORINE CONTAINING 1,4-DISUBSTITUTED PIPERIDINE DERIVATIVES, USEFUL AS ANTAGONIST FOR MUSCARINIC M3 RECEPTORS AND LESS SIDE EFFECT BANYU PHARMACEUTICAL CO LTD (JP) 2000-03-21 US disclosed
US-5948792-A POTENT AND SELECTIVE ANTAGONISTS FOR MUSCARINIC M.SUB.3 RECEPTORS WITH LITTLE SIDE EFFECTS. BANYU PHARMACEUTICAL CO., LTD. (JP) 1999-09-07 US disclosed
CN-1226888-A Fluorinated 1,4-disubstituted piperidine derivatives BANYU PHARMA CO LTD (JP) 1999-08-25 CN disclosed
EP-0930298-A1 FLUORINATED 1,4-DISUBSTITUTED PIPERIDINE DERIVATIVES BANYU PHARMACEUTICAL CO., LTD. (JP) 1999-07-21 EP disclosed