SCHEMBL7465853

SCHEMBL7465853

Fc1ccc(-c2ccc(CCBr)cc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.59
TAAR1 Q96RJ0 4/20 0.50
TDP1 Q9NUW8 1/20 0.48
IDO1 P14902 1/20 0.42
LOXL2 Q9Y4K0 1/20 0.42
AOC3 Q16853 1/20 0.42
CYP17A1 P05093 1/20 0.40
CYP21A2 P08686 1/20 0.40
CYP11B1 P15538 1/20 0.40
SIRT2 Q8IXJ6 1/20 0.40
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39
PYCR1 P32322 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL624406 0.93 TAAR1 (0.56) MAOBTAAR1TDP1IDO1LOXL2
SCHEMBL9553181 0.87 TDP1 (0.60) MAOBTAAR1TDP1
SCHEMBL9510154 0.87 TDP1 (0.60) MAOBTAAR1TDP1
Water SCHEMBL11482042 0.85 TDP1 (0.57) MAOBTAAR1TDP1
SCHEMBL9552798 0.85 MAOB (0.53) MAOBTAAR1SIRT2
SCHEMBL8015172 0.80 MAOB (0.52) MAOBTAAR1IDO1LOXL2PYCR1
SCHEMBL19651375 0.80 MAOB (0.64) MAOBTAAR1IDO1LOXL2AOC3
SCHEMBL2281085 0.79 TDP1 (0.71) MAOBTAAR1TDP1
SCHEMBL22621170 0.78 MAOB (0.61) MAOBTAAR1IDO1LOXL2
SCHEMBL22621136 0.78 MAOB (0.61) MAOBTAAR1IDO1LOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101998959-B Benzoxazole carboxamide inhibitors of poly(ADP-ribose)polymerase (PARP) BIOMARIN PHARM INC 2013-08-28 CN disclosed
CN-101998959-A Benzoxazole carboxamide inhibitors of poly(ADP-ribose)polymerase (PARP) LEAD THERAPEUTICS INC 2011-03-30 CN disclosed
EP-0837848-B1 4-ARYL-1-PHENYLALKYL-1,2,3,6-TETRAHYDROPYRIDINES HAVING NEUROTROPHIC AND NEUROPROTECTIVE ACTIVITY SANOFI SYNTHELABO (FR) 2002-09-11 EP disclosed
EP-1216996-A2 Method to synthesise biphenylyl derivatives SANOFI-SYNTHELABO (FR) 2002-06-26 EP disclosed
EP-0668286-B1 A silacyclohexane compound, a method of preparing it and a liquid crystal composition containing it SHINETSU CHEMICAL CO (JP) 2000-12-20 EP disclosed
EP-0837848-A1 4-ARYL-1-PHENYLALKYL-1,2,3,6-TETRAHYDROPYRIDINES HAVING NEUROTROPHIC AND NEUROPROTECTIVE ACTIVITY SANOFI (FR) 1998-04-29 EP disclosed
WO-1997001536-A1 4-ARYL-1-PHENYLALKYL-1,2,3,6-TETRAHYDROPYRIDINES HAVING NEUROTROPHIC AND NEUROPROTECTIVE ACTIVITY SANOFI (FR) 1997-01-16 WO disclosed
US-5523440-A Silacyclohexane compound, a method of preparaing it and a liquid crystal composition containing it SHIN-ETSU CHEMICAL CO., LTD. (JP) 1996-06-04 US disclosed
EP-0668286-A1 A silacyclohexane compound, a method of preparing it and a liquid crystal composition containing it Shin-Etsu Chemical Co., Ltd. (JP) 1995-08-23 EP disclosed