SCHEMBL7465864

SCHEMBL7465864

CCc1ccc(Nc2nccc(-c3cccn3C)n2)cc1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 6/20 0.43
KDR P35968 4/20 0.43
PTK2 Q05397 4/20 0.43
PLK1 P53350 2/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
AURKB Q96GD4 1/20 0.41
AKT1 P31749 1/20 0.41
RET P07949 3/20 0.41
JAK2 O60674 2/20 0.41
JAK3 P52333 1/20 0.41
SYK P43405 2/20 0.41
CDK4 P11802 2/20 0.41
MAPK10 P53779 1/20 0.41
CCNE1 P24864 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3517353 0.79 CDK2 (0.52) CDK2CDK4CCNE1
SCHEMBL13185630 0.78 IKBKB (0.60) PLK1NPC1RAB9AJAK2JAK3
SCHEMBL7474055 0.78 PIK3CA (0.59) CDK2KDRPTK2PLK1AURKB
SCHEMBL7460307 0.76 SYK (0.55) SYK
SCHEMBL3518870 0.76 ALDH1A1 (0.51) CDK2CDK4MAPK10
SCHEMBL3520839 0.76 CDK2 (0.52) CDK2CDK4CCNE1
SCHEMBL7465536 0.75 ABL1 (0.54) NPC1RAB9AJAK2JAK3SYK
SCHEMBL7475710 0.74 ABL1 (0.71)
SCHEMBL4159422 0.74 CDK2 (0.42) CDK2JAK2JAK3SYKCDK4
SCHEMBL7459060 0.74 NPC1 (0.46) CDK2NPC1RAB9AAURKBRET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0233461-B2 4,5,6-Substituted-2-pyrimidinamines AMERICAN CYANAMID CO (US) 2002-05-29 EP disclosed