SCHEMBL7466476

SCHEMBL7466476

CS(=O)(=O)c1ccc(-c2cc(C(F)(F)F)nn2-c2ccc(C#N)cc2)cc1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.74
CYP2C9 P11712 2/20 0.74
PTGS1 P23219 2/20 0.74
PDPK1 O15530 3/20 0.60
PTGES O14684 1/20 0.60
HDAC3 O15379 1/20 0.60
CA12 O43570 1/20 0.60
PDE5A O76074 1/20 0.60
ABCB11 O95342 1/20 0.60
MT-CO2 P00403 1/20 0.60
CA1 P00915 1/20 0.60
CA2 P00918 1/20 0.60
LMNA P02545 1/20 0.60
CA3 P07451 1/20 0.60
CYP3A4 P08684 1/20 0.60
ALOX5 P09917 1/20 0.60
ADORA3 P0DMS8 1/20 0.60
CYP2D6 P10635 1/20 0.60
ADRB3 P13945 1/20 0.60
ALOX15 P16050 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6955360 0.88 PTGS2 (0.74) PTGS2CYP2C9PTGS1PDPK1PTGES
SCHEMBL3242046 0.88 PTGS2 (0.74) PTGS2CYP2C9PTGS1PDPK1PTGES
SCHEMBL15346803 0.87 PTGS2 (0.77) PTGS2CYP2C9PTGS1PDPK1PTGES
SCHEMBL6720876 0.87 PTGS2 (0.59) PTGS2CYP2C9PTGS1PDPK1
SCHEMBL6957077 0.86 PTGS2 (0.80) PTGS2CYP2C9PTGS1PDPK1PTGES
SCHEMBL6730098 0.86 PTGS2 (0.60) PTGS2CYP2C9PTGS1PDPK1
SCHEMBL15346781 0.86 PTGS2 (0.75) PTGS2CYP2C9PTGS1PDPK1PTGES
SCHEMBL5148804 0.85 PTGS2 (0.66) PTGS2CYP2C9PTGS1PDPK1PTGES
SCHEMBL5229949 0.85 PTGS2 (1.00) PTGS2CYP2C9PTGS1PDPK1PTGES
SCHEMBL5148756 0.85 PTGS2 (0.66) PTGS2CYP2C9PTGS1PDPK1PTGES

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0554829-B1 Pyrazole derivatives with antiinflammatory, analgesic and antithrombolic activity FUJISAWA PHARMACEUTICAL CO (JP) 2002-05-15 EP disclosed
US-5670533-A ANTIINFLAMMATORY AGENTS, ANALGESICS OR ANTIRHEUMATIC DISEASES FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1997-09-23 US disclosed
US-5550147-A ANTIINFLAMMATORY AGENTS, ANALGESICS, ANTITHROMBOTIC AGENTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1996-08-27 US disclosed
EP-0554829-A2 Pyrazole derivatives with antiinflammatory, analgesic and antithrombolic activity FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-08-11 EP disclosed