SCHEMBL746937

SCHEMBL746937

COc1ccc(CC=C=O)c(OC)c1OC

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 1/20 0.45
SMN1; SMN2 Q16637 4/20 0.42
POLB P06746 2/20 0.42
CYP1A2 P05177 1/20 0.42
CHRM2 P08172 1/20 0.42
SLC6A4 P31645 1/20 0.42
OPRD1 P41143 1/20 0.42
OPRK1 P41145 1/20 0.42
KDM4E B2RXH2 6/20 0.41
TSHR P16473 1/20 0.41
APOBEC3A P31941 1/20 0.41
CTDSP1 Q9GZU7 1/20 0.41
APOBEC3G Q9HC16 1/20 0.41
ALDH1A1 P00352 5/20 0.39
MAPT P10636 2/20 0.39
LMNA P02545 2/20 0.39
GAA P10253 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
TAAR1 Q96RJ0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6606016 0.85 KDM1A (0.40) AOC3SMN1; SMN2POLBCYP1A2CHRM2
SCHEMBL5241041 0.83 ALDH1A1 (0.44) POLBKDM4ETSHRALDH1A1MAPT
SCHEMBL7151009 0.80 AOC3 (0.49) AOC3SMN1; SMN2POLBCYP1A2CHRM2
Formaldehyde SCHEMBL5244081 0.80 ALDH1A1 (0.42) POLBKDM4ETSHRALDH1A1MAPT
SCHEMBL900889 0.78 AOC3 (0.50) AOC3SMN1; SMN2POLBCYP1A2CHRM2
SCHEMBL775238 0.77 AOC3 (0.53) AOC3SMN1; SMN2POLBCYP1A2CHRM2
SCHEMBL5580537 0.77 AOC3 (0.49) AOC3SMN1; SMN2POLBCYP1A2CHRM2
SCHEMBL30883 0.75 AOC3 (0.55) AOC3SMN1; SMN2POLBCYP1A2CHRM2
SCHEMBL20573182 0.75 AOC3 (0.51) AOC3SMN1; SMN2POLBCYP1A2CHRM2
SCHEMBL27943252 0.75 AOC3 (0.44) AOC3SMN1; SMN2POLBCYP1A2CHRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2429292-A1 COMPOUNDS AND COMPOSITIONS COMPRISING CDK INHIBITORS AND METHODS FOR THE TREATMENT OF CANCER Georgia State University Research Foundation, Inc. (US) 2012-03-21 EP claimed
WO-2010129858-A1 COMPOUNDS AND COMPOSITIONS COMPRISING CDK INHIBITORS AND METHODS FOR THE TREATMENT OF CANCER GEORGIA STATE UNIVERSITY RESEARCH FOUNDATION (US) 2010-11-11 WO claimed