SCHEMBL7469620

SCHEMBL7469620

COC(=O)CCC1CCC(N2C(=O)N(c3ccc4c(c3)CCN(C(=O)C(F)(F)F)CC4)C(C)(C)C2=O)CC1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 3/20 0.38
ESR2 Q92731 3/20 0.38
NR3C2 P08235 1/20 0.35
HDAC6 Q9UBN7 2/20 0.33
FFAR4 Q5NUL3 2/20 0.31
BACE1 P56817 1/20 0.31
HDAC3 O15379 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC2 Q92769 1/20 0.31
AR P10275 1/20 0.31
ABHD6 Q9BV23 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7469615 1.00 ESR1 (0.38) ESR1ESR2NR3C2HDAC6FFAR4
SCHEMBL8564189 0.85 ESR1 (0.41) ESR1ESR2NR3C2HDAC6ABHD6
SCHEMBL8564198 0.85 ESR1 (0.41) ESR1ESR2NR3C2HDAC6ABHD6
SCHEMBL8567424 0.82 ESR1 (0.40) ESR1ESR2HDAC6ABHD6
SCHEMBL8567428 0.82 ESR1 (0.40) ESR1ESR2HDAC6ABHD6
SCHEMBL8568715 0.81 F10 (0.39) ESR1ESR2
SCHEMBL8561412 0.81 ESR1 (0.41) ESR1ESR2HDAC6ABHD6
SCHEMBL8568710 0.81 F10 (0.39) ESR1ESR2
SCHEMBL8561418 0.81 ESR1 (0.41) ESR1ESR2HDAC6ABHD6
SCHEMBL8562237 0.80 ESR1 (0.39) ESR1ESR2HDAC6BACE1ABHD6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0777667-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT Dr. Karl Thomae GmbH (DE) 1997-06-11 EP disclosed
WO-1996005194-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT DR. KARL THOMAE GMBH (DE) 1996-02-22 WO disclosed