SCHEMBL8564198

SCHEMBL8564198

COC(=O)CCC1CCC(N2C(=O)CN(c3ccc4c(c3)CCN(C(=O)C(F)(F)F)CC4)C2=O)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 4/20 0.41
ESR2 Q92731 4/20 0.41
HDAC6 Q9UBN7 2/20 0.34
ABHD6 Q9BV23 1/20 0.33
NR3C2 P08235 1/20 0.33
PDE4B Q07343 1/20 0.32
PDE4D Q08499 1/20 0.32
HTR1A P08908 2/20 0.32
DRD3 P35462 2/20 0.32
HDAC8 Q9BY41 1/20 0.32
TMEM97 Q5BJF2 4/20 0.31
SIGMAR1 Q99720 4/20 0.31
TYRO3 Q06418 1/20 0.31
MERTK Q12866 1/20 0.31
KDM4E B2RXH2 1/20 0.31
CHRM4 P08173 1/20 0.31
CHRM5 P08912 1/20 0.31
ADRA2A P08913 1/20 0.31
ADRA2B P18089 1/20 0.31
HRH2 P25021 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8564189 1.00 ESR1 (0.41) ESR1ESR2HDAC6ABHD6NR3C2
SCHEMBL8567424 0.87 ESR1 (0.40) ESR1ESR2HDAC6ABHD6DRD3
SCHEMBL8567428 0.87 ESR1 (0.40) ESR1ESR2HDAC6ABHD6DRD3
SCHEMBL8568710 0.86 F10 (0.39) ESR1ESR2
SCHEMBL8561412 0.86 ESR1 (0.41) ESR1ESR2HDAC6ABHD6PDE4B
SCHEMBL8568715 0.86 F10 (0.39) ESR1ESR2
SCHEMBL8561418 0.86 ESR1 (0.41) ESR1ESR2HDAC6ABHD6PDE4B
SCHEMBL7469615 0.85 ESR1 (0.38) ESR1ESR2HDAC6ABHD6NR3C2
SCHEMBL7469620 0.85 ESR1 (0.38) ESR1ESR2HDAC6ABHD6NR3C2
Hydrochloric Acid SCHEMBL8595133 0.84 HTR6 (0.39) HTR1ADRD3HTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0612741-B1 Cyclic derivatives, medicaments containing them and process for their preparation THOMAE GMBH DR K (DE) 1998-06-10 EP disclosed
US-5612335-A ANTICOAGULANTS; COMBATING/PREVENTING DISEASES WHERE CELL AGGREGATES OCCUR OR CELL-MATRIX INTERACTIONS PLAY A PART KARL THOMAE GMBH (DE) 1997-03-18 US disclosed
US-5519036-A IMIDAZOLIDINONES, ANTICOAGULANTS, CELL AGGREGATION PREVENTION KARL THOMAE GMBH (DE) 1996-05-21 US disclosed
EP-0612741-A1 Cyclic derivatives, medicaments containing them and process for their preparation Dr. Karl Thomae GmbH (DE) 1994-08-31 EP disclosed