SCHEMBL7470255

SCHEMBL7470255

CCN(CC)C(=O)Nc1ccc(S(=O)(=O)N2C(=O)C(NCCCCCN)(c3ccccc3Cl)c3cc(Cl)c(Cl)cc32)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.35
GAA P10253 1/20 0.35
CA12 O43570 2/20 0.34
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
CA9 Q16790 2/20 0.34
GHSR Q92847 2/20 0.32
LMNA P02545 2/20 0.32
MAPT P10636 2/20 0.32
NAMPT P43490 1/20 0.32
NR1I3 Q14994 1/20 0.31
MERTK Q12866 1/20 0.31
ALDH1A1 P00352 2/20 0.31
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 2/20 0.30
KMT2A Q03164 2/20 0.30
TP53 P04637 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL8589290 0.95 CACNA1B (0.36) NPSR1GAACA12CA1CA2
SCHEMBL7471274 0.93 NPSR1 (0.38) NPSR1GAACA12CA1CA2
SCHEMBL7477246 0.92 NPSR1 (0.39) NPSR1GAACA12CA1CA2
Trifluoroacetic Acid SCHEMBL8592809 0.88 NPSR1 (0.36) NPSR1GAACA12CA1CA2
SCHEMBL7476887 0.85 NPSR1 (0.39) NPSR1GAACA12CA1CA2
SCHEMBL7471149 0.84 NPSR1 (0.39) NPSR1GAACA12CA1CA2
SCHEMBL236066 0.83 NPSR1 (0.33) NPSR1GAAMAPTNAMPTNR1I3
SCHEMBL7472360 0.83 NPSR1 (0.38) NPSR1GAACA12CA1CA2
SCHEMBL8742735 0.83 NPSR1 (0.40) NPSR1GAACA12CA1CA2
SCHEMBL7471625 0.82 NPSR1 (0.41) NPSR1GAACA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0687251-B1 1,3-DIHYDROINDOL-2-ONE DERIVATIVES SUBSTITUTED IN POSITION 3 BY A NITROGEN GROUP AS VASOPRESSIN AND/OR OCYTOCINE AGONISTS AND/OR ANTAGONISTS SANOFI SYNTHELABO (FR) 2002-02-27 EP disclosed
EP-0687251-A1 1,3-DIHYDROINDOL-2-ONE DERIVATIVES SUBSTITUTED IN POSITION 3 BY A NITROGEN GROUP AS VASOPRESSIN AND/OR OCYTOCINE AGONISTS AND/OR ANTAGONISTS SANOFI (FR) 1995-12-20 EP disclosed
WO-1995018105-A1 1,3-DIHYDROINDOL-2-ONE DERIVATIVES SUBSTITUTED IN POSITION 3 BY A NITROGEN GROUP AS VASOPRESSIN AND/OR OCYTOCINE AGONISTS AND/OR ANTAGONISTS SANOFI (FR) 1995-07-06 WO disclosed