SCHEMBL7470485

SCHEMBL7470485

CN1CCc2ccc(N3CCN(CCC(=O)NCCC(=O)O)C3=O)cc2CC1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.45
ITGB3 P05106 5/20 0.44
ITGA2B P08514 5/20 0.44
DRD3 P35462 5/20 0.39
KCNH2 Q12809 4/20 0.39
DRD2 P14416 4/20 0.39
HDAC1 Q13547 3/20 0.37
DPP4 P27487 4/20 0.36
DPP8 Q6V1X1 2/20 0.36
GRIN1 Q05586 1/20 0.35
GRIN2B Q13224 1/20 0.35
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
POLB P06746 1/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7474275 0.92 ITGB3 (0.51) S1PR1ITGB3ITGA2BDRD3KCNH2
SCHEMBL7467606 0.91 S1PR1 (0.43) S1PR1ITGB3ITGA2BDRD3KCNH2
SCHEMBL7472620 0.90 ITGB3 (0.49) S1PR1ITGB3ITGA2BHDAC1
Hydrochloric Acid SCHEMBL7420584 0.88 S1PR1 (0.54) S1PR1DRD3KCNH2DRD2HDAC1
SCHEMBL7479149 0.87 ITGB3 (0.40) S1PR1ITGB3ITGA2BDRD3KCNH2
SCHEMBL7481405 0.87 NR1H2 (0.42) S1PR1ITGB3ITGA2BMEN1POLB
SCHEMBL7483682 0.82 DRD3 (0.40) S1PR1DRD3KCNH2DRD2HDAC1
Hydrochloric Acid SCHEMBL7472463 0.80 DRD3 (0.42) S1PR1DRD3KCNH2DRD2HDAC1
Hydrochloric Acid SCHEMBL8557146 0.80 S1PR1 (0.53) S1PR1DRD3KCNH2DRD2HDAC1
SCHEMBL7481505 0.79 DRD3 (0.41) S1PR1DRD3KCNH2DRD2HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0777667-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT Dr. Karl Thomae GmbH (DE) 1997-06-11 EP disclosed
WO-1996005194-A1 CYCLIC BENZAZEPINE UREA DERIVATIVES WITH AGGREGATION-INHIBITING EFFECT DR. KARL THOMAE GMBH (DE) 1996-02-22 WO disclosed