SCHEMBL7471145

SCHEMBL7471145

Nc1ccc(N)c(-c2nccc(-c3cccnc3)n2)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.57
HSP90AB1 P08238 1/20 0.57
PTK2 Q05397 1/20 0.57
ABL1 P00519 9/20 0.54
BCR P11274 8/20 0.54
EGFR P00533 3/20 0.54
SRC P12931 2/20 0.54
PRKACA P17612 1/20 0.54
PRKACG P22612 1/20 0.54
PRKACB P22694 1/20 0.54
ABL2 P42684 1/20 0.47
MEN1 O00255 1/20 0.46
PSIP1 O75475 1/20 0.46
AXL P30530 1/20 0.46
MKNK1 Q9BUB5 1/20 0.46
MKNK2 Q9HBH9 1/20 0.46
PRKCA P17252 4/20 0.45
PRKCD Q05655 2/20 0.45
CYP2A6 P11509 2/20 0.44
LOXL2 Q9Y4K0 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30921140 1.00 HSP90AA1 (0.57) HSP90AA1HSP90AB1PTK2ABL1BCR
SCHEMBL22206280 0.86 ABL1 (0.63) HSP90AA1HSP90AB1PTK2ABL1BCR
Ammonia Solution, Strong SCHEMBL2693849 0.85 ABL1 (0.62) HSP90AA1HSP90AB1PTK2ABL1BCR
Hydrochloric Acid SCHEMBL5531500 0.84 ABL1 (0.61) HSP90AA1HSP90AB1PTK2ABL1BCR
SCHEMBL7476653 0.82 ABL1 (0.48) HSP90AA1ABL1BCREGFRSRC
SCHEMBL145074 0.80 AXL (0.59) MEN1PSIP1AXLMKNK1MKNK2
Hydrochloric Acid SCHEMBL6739740 0.79 AXL (0.58) MEN1PSIP1AXLMKNK1MKNK2
Hydrochloric Acid SCHEMBL7090061 0.79 AXL (0.58) MEN1PSIP1AXLMKNK1MKNK2
SCHEMBL207818 0.77 CYP19A1 (0.64) AXLMKNK1MKNK2MAPTCYP19A1
SCHEMBL1231783 0.77 HSP90AA1 (0.64) HSP90AA1HSP90AB1PTK2ABL1BCR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0233461-B2 4,5,6-Substituted-2-pyrimidinamines AMERICAN CYANAMID CO (US) 2002-05-29 EP disclosed
EP-0233461-B1 4,5,6-Substituted-2-pyrimidinamines AMERICAN CYANAMID CO (US) 1996-03-20 EP disclosed