SCHEMBL7471573

SCHEMBL7471573

c1ccc(N2CCC(CNCC3COc4ccccc4O3)CC2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 12/20 1.00
ADRA1A P35348 12/20 1.00
ADRA1B P35368 12/20 1.00
ALDH1A1 P00352 1/20 0.56
HPGD P15428 1/20 0.56
HTR1A P08908 1/20 0.55
DRD2 P14416 1/20 0.55
DRD4 P21917 1/20 0.55
HTR2C P28335 1/20 0.55
DRD3 P35462 1/20 0.55
POLB P06746 1/20 0.52
ESR2 Q92731 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8124825 0.99 ADRA1D (0.98) ADRA1DADRA1AADRA1BALDH1A1HPGD
SCHEMBL7466659 0.88 ADRA1D (1.00) ADRA1DADRA1AADRA1BALDH1A1HTR1A
Hydrochloric Acid SCHEMBL8127001 0.87 ADRA1D (0.98) ADRA1DADRA1AADRA1BALDH1A1HTR1A
SCHEMBL7464233 0.86 ADRA1D (1.00) ADRA1DADRA1AADRA1BHTR1ADRD2
SCHEMBL7473727 0.85 ADRA1D (1.00) ADRA1DADRA1AADRA1BALDH1A1HPGD
Hydrochloric Acid SCHEMBL8118058 0.85 ADRA1D (0.98) ADRA1DADRA1AADRA1BHTR1ADRD2
Hydrochloric Acid SCHEMBL8131921 0.84 ADRA1D (0.98) ADRA1DADRA1AADRA1BALDH1A1HPGD
SCHEMBL7463873 0.82 ADRA1D (0.80) ADRA1DADRA1AADRA1B
Hydrochloric Acid SCHEMBL7459565 0.82 ADRA1D (0.78) ADRA1DADRA1AADRA1B
SCHEMBL7466851 0.82 ADRA1D (1.00) ADRA1DADRA1AADRA1BALDH1A1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1198234-A2 BICYCLIC AROMATIC COMPOUNDS FOR TREATING DRUG ADDICTION Knoll GmbH (DE) 2002-04-24 EP claimed
WO-2001002391-A2 BICYCLIC AROMATIC COMPOUNDS FOR TREATING DRUG ADDICTION KNOLL GMBH (DE) 2001-01-11 WO claimed
CN-1052723-C Bicyclic aromatic compounds as therapeutic agents KNOLL AG (DE) 2000-05-24 CN claimed
EP-0717739-B1 1,4-Benzodioxane derivatives having affinity for D2 receptors and utility in the treatment of psychoses KNOLL AG (DE) 2000-03-29 EP claimed
CN-1133043-A Bicyclic aromatic compounds as therapeutic agents BOOTS CO PLC (DE) 1996-10-09 CN claimed
EP-0717739-A1 BICYCLIC AROMATIC COMPOUNDS AS THERAPEUTIC AGENTS Knoll AG (DE) 1996-06-26 EP claimed
WO-1995007274-A1 BICYCLIC AROMATIC COMPOUNDS AS THERAPEUTIC AGENTS KNOLL AG (DE) 1995-03-16 WO claimed
EP-1198234-A2 BICYCLIC AROMATIC COMPOUNDS FOR TREATING DRUG ADDICTION Knoll GmbH (DE) 2002-04-24 EP disclosed
WO-2001002391-A2 BICYCLIC AROMATIC COMPOUNDS FOR TREATING DRUG ADDICTION KNOLL GMBH (DE) 2001-01-11 WO disclosed
CN-1052723-C Bicyclic aromatic compounds as therapeutic agents KNOLL AG (DE) 2000-05-24 CN disclosed
EP-0717739-B1 1,4-Benzodioxane derivatives having affinity for D2 receptors and utility in the treatment of psychoses KNOLL AG (DE) 2000-03-29 EP disclosed
US-5767116-A TREATING PSYCHOSES KNOLL ATKIENGESELLSCHAFT (DE) 1998-06-16 US disclosed
CN-1133043-A Bicyclic aromatic compounds as therapeutic agents BOOTS CO PLC (DE) 1996-10-09 CN disclosed