SCHEMBL7472203

SCHEMBL7472203

NN(c1ccc(-c2ccccc2)cc1)C1CCCCC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH4 Q9H3N8 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40
ENPP2 Q13822 1/20 0.39
MCL1 Q07820 1/20 0.39
KDM4E B2RXH2 2/20 0.38
MEN1 O00255 2/20 0.38
ALDH1A1 P00352 2/20 0.38
KMT2A Q03164 2/20 0.38
NPC1 O15118 1/20 0.38
MITF O75030 1/20 0.38
RAB9A P51151 1/20 0.38
PAX8 Q06710 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PTGES O14684 1/20 0.37
ALOX5 P09917 1/20 0.37
GPR88 Q9GZN0 2/20 0.37
S1PR1 P21453 1/20 0.36
S1PR3 Q99500 1/20 0.36
KDM1A O60341 2/20 0.36
MAOB P27338 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18639248 0.88 KDM4E (0.46) KDM4EMEN1ALDH1A1KMT2ANPC1
SCHEMBL5971405 0.88 KDM4E (0.46) KDM4EMEN1ALDH1A1KMT2ANPC1
Hydrochloric Acid SCHEMBL9391758 0.86 KDM4E (0.45) KDM4EMEN1ALDH1A1KMT2ANPC1
Hydrochloric Acid SCHEMBL7818342 0.86 KDM4E (0.45) KDM4EMEN1ALDH1A1KMT2ANPC1
SCHEMBL3485394 0.86 KDM4E (0.43) KDM4EMEN1ALDH1A1KMT2ANPC1
SCHEMBL8518648 0.78 TAAR1 (0.36) KDM4EMEN1ALDH1A1KMT2ANPC1
SCHEMBL14817427 0.77 KCNA3 (0.48) HRH4HRH3ENPP2MCL1KDM4E
Hydrochloric Acid SCHEMBL28010546 0.76 TAAR1 (0.35) KDM4EMEN1ALDH1A1KMT2ANPC1
SCHEMBL10793012 0.75 MCL1 (0.43) HRH4HRH3ENPP2MCL1KDM4E
SCHEMBL25987505 0.75 KCNA3 (0.43) HRH4HRH3ENPP2MCL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1058678-B1 METAL-CATALYZED ARYLATIONS AND VINYLATIONS OF HYDRAZINES, HYDRAZONES, HYDROXYLAMINES AND OXIMES MASSACHUSETTS INST TECHNOLOGY (US) 2002-12-11 EP disclosed
US-6465693-B2 TRANSITION METAL CATALYZED ARYLATION OR VINYLATION; COMBINATORIAL CHEMISTRY MASSACHUSETTS INSTITUTE OF TECHNOLOGY 2002-10-15 US disclosed
US-20010031894-A1 Metal-catalyzed arylations of hydrazines, hydrazones, and related substrates BUCHWALD STEPHEN L (US) 2001-10-18 US disclosed
US-6235936-B1 TRANSITION METAL CATALYST FOR ARYLATION MASSACHUSETTS INSTITUTE OF TECHNOLOGY 2001-05-22 US disclosed
EP-1058678-A2 METAL-CATALYZED ARYLATIONS AND VINYLATIONS OF HYDRAZINES, HYDRAZONES, HYDROXYLAMINES AND OXIMES Massachusetts Institute of Technology (US) 2000-12-13 EP disclosed
WO-1999043643-A2 METAL-CATALYZED ARYLATIONS AND VINYLATIONS OF HYDRAZINES, HYDRAZONES, HYDROXYLAMINES AND OXIMES MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 1999-09-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010031894-A1 Metal-catalyzed arylations of hydrazines, hydrazones, and related substrates IDO1, IDO2, AHR HRH4 401/4885HRH3 724/4885ENPP2 3153/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.