SCHEMBL7474047

SCHEMBL7474047

O=C(c1ccccn1)c1nsc2nccn12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.46
CES2 O00748 1/20 0.43
CES1 P23141 1/20 0.43
L3MBTL1 Q9Y468 3/20 0.42
LMNA P02545 3/20 0.42
NAPRT Q6XQN6 1/20 0.42
P4HTM Q9NXG6 1/20 0.42
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 2/20 0.40
GSK3B P49841 1/20 0.38
HSD17B14 Q9BPX1 1/20 0.38
MAPT P10636 1/20 0.37
F13A1 P00488 1/20 0.37
RAB9A P51151 3/20 0.37
NPC1 O15118 2/20 0.37
PKM P14618 1/20 0.37
SMYD3 Q9H7B4 1/20 0.36
CA1 P00915 2/20 0.36
CA2 P00918 2/20 0.36
CA4 P22748 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7473176 0.73 F13A1 (0.38) KMT2AALDH1A1KDM4EF13A1
SCHEMBL7479423 0.72 KDM4E (0.46) KMT2ACES2CES1L3MBTL1LMNA
SCHEMBL87791 0.71 KMT2A (0.75) KMT2ACES2CES1L3MBTL1LMNA
SCHEMBL31369148 0.71 KMT2A (0.75) KMT2ACES2CES1L3MBTL1LMNA
SCHEMBL7533418 0.70 TDP1 (0.45) KMT2AL3MBTL1LMNAALDH1A1KDM4E
Charcoal, Activated SCHEMBL8358164 0.69 KMT2A (0.72) KMT2ACES2CES1L3MBTL1LMNA
Hydrochloric Acid SCHEMBL27723543 0.69 KMT2A (0.72) KMT2ACES2CES1L3MBTL1LMNA
Water SCHEMBL6228901 0.69 KMT2A (0.72) KMT2ACES2CES1L3MBTL1LMNA
SCHEMBL31369119 0.69 KMT2A (0.72) KMT2ACES2CES1L3MBTL1LMNA
SCHEMBL24977120 0.66 KMT2A (0.67) KMT2ACES2CES1L3MBTL1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0883622-B1 PROTON PUMP INHIBITOR APOTEX INC (CA) 2002-05-15 EP disclosed
US-6114537-A 1,2,4-THIADIAZOLE COMPOUND IS USEFUL FOR TRAPPING THIOL COMPOUNDS AND SELECTIVELY CHANGING THIOLS TO DISULFIDE COMPOUNDS APOTEX INC. (CA) 2000-09-05 US disclosed
US-6093738-A IMIDAZO(1,2-D)-THIADIAZOLE COMPOUNDS; PEPTIC ULCER TREATMENT KARIMIAN KHASHAYAR (CA) 2000-07-25 US disclosed
EP-0883622-A1 PROTON PUMP INHIBITOR APOTEX INC. (CA) 1998-12-16 EP disclosed
WO-1997031923-A1 PROTON PUMP INHIBITOR APOTEX INC. (CA) 1997-09-04 WO disclosed