SCHEMBL7474749

SCHEMBL7474749

Nc1[nH]nc(-c2ccc(F)cc2)c1C(=O)c1cccc(CN2CCCCC2)c1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
HIF1A Q16665 1/20 0.49
ALDH1A1 P00352 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
CSNK1D P48730 2/20 0.43
DYRK1A Q13627 4/20 0.43
CSNK1E P49674 1/20 0.43
PTPN2 P17706 1/20 0.42
GRM2 Q14416 1/20 0.42
WNT1 P04628 3/20 0.42
HTR2C P28335 1/20 0.41
MCHR1 Q99705 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7475964 0.88 CYP2D6 (0.47) CYP2D6CYP2C9HIF1AALDH1A1SMN1; SMN2
SCHEMBL7474456 0.81 MAPK14 (0.52)
SCHEMBL1383396 0.81 MAPK14 (0.52)
SCHEMBL7803286 0.81 MAPK14 (0.54) CYP2D6
Hydrochloric Acid SCHEMBL7473782 0.81 MAPK14 (0.51)
SCHEMBL5322574 0.80 MAPK14 (0.61) ALDH1A1DYRK1AWNT1
SCHEMBL7476872 0.80 MAPK14 (0.45)
SCHEMBL1385251 0.79 MAPK14 (0.55)
Hydrochloric Acid SCHEMBL7468024 0.79 MAPK14 (0.60) DYRK1AWNT1
SCHEMBL1383366 0.79 MAPK14 (0.57)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218346-A1 PYRAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-07-03 EP disclosed
WO-2001021591-A1 PYRAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2001-03-29 WO disclosed