SCHEMBL7475524

SCHEMBL7475524

[CH2]c1ccc(OC)cc1C(=O)NO

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.53
CA2 P00918 1/20 0.53
MMP2 P08253 3/20 0.46
MMP9 P14780 3/20 0.46
MMP8 P22894 3/20 0.46
MMP12 P39900 3/20 0.46
MMP13 P45452 3/20 0.46
MMP14 P50281 3/20 0.46
MMP16 P51512 3/20 0.46
KDM4E B2RXH2 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2D6 P10635 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
MAPT P10636 1/20 0.44
HTT P42858 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
HDAC8 Q9BY41 3/20 0.43
HPGD P15428 2/20 0.43
NPC1 O15118 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1436731 0.81 P2RX1 (0.57) CA1CA2KDM4ECYP1A2CYP2C19
SCHEMBL8483740 0.80 SMN1; SMN2 (0.59) CA1CA2KDM4EMAPTHTT
SCHEMBL16495950 0.78 CA1 (0.51) CA1CA2MMP2MMP9MMP8
SCHEMBL1562332 0.77 NPC1 (0.68) CA1CA2CYP1A2CYP2D6CYP2C19
SCHEMBL16958941 0.71 KDM4E (0.56) CA1CA2KDM4ECYP1A2CYP2D6
SCHEMBL976321 0.70 MEN1 (0.48) KDM4EMAPTNPSR1HDAC8HPGD
SCHEMBL10839189 0.70 CA1 (0.70) CA1CA2KDM4EHDAC8NPC1
SCHEMBL942259 0.70 CA1 (1.00) CA1CA2CYP1A2CYP2D6CYP2C9
SCHEMBL8478835 0.69 SMN1; SMN2 (0.54) CA1CA2KDM4EHPGDNPC1
SCHEMBL7502111 0.69 HPGD (0.61) KDM4ECYP1A2CYP2C19MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6482827-B1 Matrix metalloproteinase inhibitors PHARMACIA & UPJOHN S.P.A. (IT) 2002-11-19 US disclosed
EP-0925289-A1 MATRIX METALLOPROTEINASE INHIBITORS PHARMACIA & UPJOHN S.p.A. (IT) 1999-06-30 EP disclosed
WO-1999002510-A1 MATRIX METALLOPROTEINASE INHIBITORS PHARMACIA & UPJOHN S.P.A. (IT) 1999-01-21 WO disclosed