SCHEMBL7475909

SCHEMBL7475909

C=C[CH]c1cccc(F)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 11/20 0.60
CYP1A2 P05177 1/20 0.54
CYP3A4 P08684 1/20 0.54
CYP2D6 P10635 1/20 0.54
PKM P14618 1/20 0.54
MAPK1 P28482 1/20 0.54
THPO P40225 1/20 0.54
NPC1 O15118 1/20 0.54
CHRM5 P08912 1/20 0.54
GRM5 P41594 1/20 0.54
RAB9A P51151 1/20 0.54
BLM P54132 1/20 0.54
PMP22 Q01453 1/20 0.54
PTGS1 P23219 3/20 0.47
PTGS2 P35354 1/20 0.47
NQO2 P16083 1/20 0.46
FBP1 P09467 1/20 0.44
RELA Q04206 1/20 0.43
IKBKB O14920 1/20 0.42
FGFR1 P11362 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29694491 0.81
SCHEMBL49997 0.81
Hydrogen Sulfide SCHEMBL31655513 0.79 NFE2L2 (0.62) NFE2L2CYP1A2CYP3A4CYP2D6PKM
SCHEMBL29108870 0.78 NFE2L2 (0.68) NFE2L2CYP1A2CYP3A4CYP2D6PKM
SCHEMBL19540032 0.78 NFE2L2 (0.68) NFE2L2CYP1A2CYP3A4CYP2D6PKM
SCHEMBL18255133 0.78 NFE2L2 (0.68) NFE2L2CYP1A2CYP3A4CYP2D6PKM
SCHEMBL1759769 0.77 NFE2L2 (0.60) NFE2L2CYP1A2CYP3A4CYP2D6PKM
Cyanide SCHEMBL28745996 0.76 NFE2L2 (0.58) NFE2L2CYP1A2CYP3A4CYP2D6PKM
SCHEMBL31317689 0.75 NFE2L2 (1.00) NFE2L2CYP1A2CYP3A4CYP2D6PKM
SCHEMBL700536 0.75 NFE2L2 (1.00) NFE2L2CYP1A2CYP3A4CYP2D6PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2900645-A1 3-PHENYLISOXAZOLIN DERIVATIVES WITH HERBICIDAL ACTION Bayer CropScience AG (DE) 2015-08-05 EP disclosed
EP-0742218-B1 PYRROLOPYRIDAZINE DERIVATIVE SANKYO CO (JP) 2002-12-04 EP disclosed
US-6063782-A Pyrrolopyridazine derivatives SANKYO COMPANY, LIMITED (JP) 2000-05-16 US disclosed
CN-1143964-A Pyrrolopyridazine derivative SANKYO CO (JP) 1997-02-26 CN disclosed
EP-0742218-A1 PYRROLOPYRIDAZINE DERIVATIVE SANKYO COMPANY LIMITED (JP) 1996-11-13 EP disclosed