SCHEMBL7477116

SCHEMBL7477116

CC(C)(C)[Si](C)(C)Oc1ccc(C2C(=O)NC(=O)NC2=O)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PREP P48147 4/20 0.46
CA12 O43570 4/20 0.44
CA1 P00915 4/20 0.44
CA9 Q16790 4/20 0.44
ALDH1A1 P00352 3/20 0.35
MAPT P10636 2/20 0.35
LMNA P02545 2/20 0.34
ABL1 P00519 1/20 0.33
KMT2A Q03164 1/20 0.33
RIN1 Q13671 1/20 0.33
HAO1 Q9UJM8 1/20 0.33
HPGD P15428 2/20 0.31
KDM4E B2RXH2 2/20 0.31
GAA P10253 1/20 0.31
HSD17B10 Q99714 1/20 0.31
TP53 P04637 2/20 0.31
NPC1 O15118 1/20 0.31
MAOA P21397 1/20 0.31
PTGS2 P35354 1/20 0.31
RAB9A P51151 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7477778 0.83 CA12 (0.41) PREPCA12CA1CA9ALDH1A1
SCHEMBL6385836 0.75 HPGD (0.53) CA12CA1CA9ALDH1A1MAPT
SCHEMBL6763899 0.74 PREP (0.53) PREPCA12CA1CA9ALDH1A1
SCHEMBL30830698 0.73 CRBN (0.64) PREPNPC1DDB1CRBN
SCHEMBL7480650 0.73 PREP (0.46) PREPCA12CA1CA9LMNA
SCHEMBL28843306 0.71 CA12 (0.41) PREPCA12CA1CA9
SCHEMBL28843303 0.71 CA12 (0.41) PREPCA12CA1CA9
SCHEMBL6437309 0.70 ESR2 (0.47) PREPCA12CA1CA9ALDH1A1
SCHEMBL20640939 0.70 PREP (0.43) PREPCA12CA1CA9DDB1
SCHEMBL29223877 0.70 CA12 (0.42) PREPCA12CA1CA9MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6472396-B1 Barbituric acid derivatives, processes for their production and pharmaceutical agents containing these compounds ROCHE DIAGNOSTICS GMBH (DE) 2002-10-29 US disclosed
EP-0869947-B1 BARBITURIC ACID DERIVATIVES, PROCESSES FOR THEIR PRODUCTION AND PHARMACEUTICAL AGENTS CONTAINING THESE COMPOUNDS ROCHE DIAGNOSTICS GMBH (DE) 2002-10-23 EP disclosed
US-6110924-A MATRIX METALLOPROTEASE INHIBITORS ROCHE DIAGNOSTICS GMBH (DE) 2000-08-29 US disclosed
EP-0869947-A1 NEW BARBITURIC ACID DERIVATIVES, PROCESSES FOR THEIR PRODUCTION AND PHARMACEUTICAL AGENTS CONTAINING THESE COMPOUNDS Roche Diagnostics GmbH (DE) 1998-10-14 EP disclosed
WO-1997023465-A1 NEW BARBITURIC ACID DERIVATIVES, PROCESSES FOR THEIR PRODUCTION AND PHARMACEUTICAL AGENTS CONTAINING THESE COMPOUNDS BOEHRINGER MANNHEIM GMBH (DE) 1997-07-03 WO disclosed