SCHEMBL7477188

SCHEMBL7477188

CC1(C)C(=O)Nc2c(Cl)cccc2C1=O

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NSD2 O96028 2/20 0.53
BCHE P06276 1/20 0.53
DAO P14920 1/20 0.53
CES1 P23141 1/20 0.53
TGM2 P21980 2/20 0.45
TYMS P04818 1/20 0.43
PDK2 Q15119 4/20 0.41
MAPT P10636 4/20 0.41
PDK4 Q16654 3/20 0.40
PDK1 Q15118 1/20 0.40
PDK3 Q15120 1/20 0.40
AHR P35869 1/20 0.40
PKM P14618 1/20 0.38
KDM4E B2RXH2 2/20 0.38
BLM P54132 2/20 0.38
MEN1 O00255 1/20 0.38
ALDH1A1 P00352 1/20 0.38
TP53 P04637 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7423435 0.79 CA1 (0.43) DAOTGM2TYMSPDK2MAPT
SCHEMBL7484503 0.78 NSD2 (0.49) NSD2BCHEDAOCES1TGM2
SCHEMBL2269040 0.78 PDK2 (0.61) NSD2BCHEDAOCES1TGM2
SCHEMBL7479441 0.76 CA1 (0.45) TYMSPDK2MAPTPDK4PDK1
SCHEMBL7478070 0.75 NSD2 (0.42) NSD2BCHEDAOCES1TGM2
SCHEMBL7472238 0.75 NSD2 (0.42) NSD2BCHEDAOCES1TGM2
SCHEMBL7483462 0.75 NSD2 (0.42) NSD2BCHEDAOCES1TGM2
SCHEMBL25112387 0.72 CES1 (0.77) NSD2BCHEDAOCES1TGM2
SCHEMBL2818017 0.72 TYMS (0.52) NSD2BCHEDAOCES1TGM2
SCHEMBL19855787 0.69 CES1 (0.71) NSD2BCHEDAOCES1TGM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0697405-B1 Substituted quinoline derivatives, process for their preparation and their use AVENTIS PHARMA GMBH (DE) 2002-08-14 EP disclosed
EP-0579968-B1 4-Iminoquinolines, processes for their preparation and their use HOECHST AG (DE) 1999-09-01 EP disclosed
EP-0697405-A1 Substituted quinoline derivatives, process for their preparation and their use HOECHST AKTIENGESELLSCHAFT (DE) 1996-02-21 EP disclosed
EP-0579968-A1 4-Iminoquinolines, processes for their preparation and their use HOECHST AKTIENGESELLSCHAFT (DE) 1994-01-26 EP disclosed