SCHEMBL7477768

SCHEMBL7477768

C/C=C/Cn1c(C)c(C)c2cnnc(SCc3ccc(Cl)cc3Cl)c21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.40
CYP1A2 P05177 5/20 0.38
CYP2C19 P33261 5/20 0.38
HPGD P15428 4/20 0.37
NPSR1 Q6W5P4 3/20 0.37
TSHR P16473 1/20 0.37
KMT2A Q03164 2/20 0.36
CA5A P35218 1/20 0.36
ALDH1A1 P00352 3/20 0.36
MCL1 Q07820 1/20 0.36
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TP53 P04637 2/20 0.34
HTT P42858 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
EGFR P00533 1/20 0.34
MET P08581 1/20 0.34
CYP3A4 P08684 4/20 0.33
CYP2C9 P11712 4/20 0.33
CYP2D6 P10635 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7477772 1.00 MAPT (0.40) MAPTCYP1A2CYP2C19HPGDNPSR1
SCHEMBL7477360 0.82 PTK2 (0.33) CYP1A2CYP2C19RAB9ASMN1; SMN2TP53
SCHEMBL7477363 0.82 PTK2 (0.33) CYP1A2CYP2C19RAB9ASMN1; SMN2TP53
SCHEMBL7477837 0.80 CYP1A2 (0.41) MAPTCYP1A2CYP2C19HPGDNPSR1
SCHEMBL7477834 0.80 CYP1A2 (0.41) MAPTCYP1A2CYP2C19HPGDNPSR1
SCHEMBL7479365 0.79 MEN1 (0.40) MAPTCYP1A2CYP2C19NPSR1TSHR
SCHEMBL7479371 0.79 MEN1 (0.40) MAPTCYP1A2CYP2C19NPSR1TSHR
SCHEMBL7478254 0.78 CYP1A2 (0.41) MAPTCYP1A2CYP2C19HPGDNPSR1
SCHEMBL7478248 0.78 CYP1A2 (0.41) MAPTCYP1A2CYP2C19HPGDNPSR1
SCHEMBL7483941 0.76 L3MBTL1 (0.37) MAPTTSHRKMT2AALDH1A1MCL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0742218-B1 PYRROLOPYRIDAZINE DERIVATIVE SANKYO CO (JP) 2002-12-04 EP disclosed
US-6063782-A Pyrrolopyridazine derivatives SANKYO COMPANY, LIMITED (JP) 2000-05-16 US disclosed
EP-0742218-A1 PYRROLOPYRIDAZINE DERIVATIVE SANKYO COMPANY LIMITED (JP) 1996-11-13 EP disclosed