SCHEMBL7477884

SCHEMBL7477884

CCc1nc2ccc(O)cc2n1C(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 1/20 0.39
ESR2 Q92731 3/20 0.39
NR1H2 P55055 8/20 0.37
NR1H3 Q13133 3/20 0.35
ESR1 P03372 2/20 0.35
ACSS2 Q9NR19 1/20 0.35
GABRG2 P18507 1/20 0.34
GABRB3 P28472 1/20 0.34
GABRA5 P31644 1/20 0.34
ESRRB O95718 1/20 0.34
ESRRA P11474 1/20 0.34
RPS6KA5 O75582 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7473742 0.90 CNR2 (0.41) HTR6ESR2NR1H2NR1H3ESR1
SCHEMBL7486828 0.88 CNR2 (0.43) HTR6ESR2NR1H2ESR1
SCHEMBL7482600 0.86 CNR2 (0.41) HTR6ESR2NR1H2NR1H3
SCHEMBL7476588 0.84 HTR6 (0.38) HTR6ESR2NR1H2NR1H3
SCHEMBL23448942 0.83 HTR6 (0.35) HTR6ESR2NR1H2NR1H3
SCHEMBL14300652 0.83 CYP1A2 (0.46) NR1H2NR1H3
SCHEMBL7480954 0.83 ESR2 (0.41) HTR6ESR2NR1H2NR1H3GABRG2
SCHEMBL7483480 0.82 CNR2 (0.41) HTR6ESR2NR1H2NR1H3ACSS2
SCHEMBL7482978 0.80 ESR2 (0.39) HTR6ESR2NR1H2ACSS2GABRG2
SCHEMBL7486188 0.80 CNR2 (0.39) HTR6ESR2NR1H2NR1H3ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0865281-B1 NAPHTHYL-SUBSTITUTED BENZIMIDAZOLE DERIVATIVES AS ANTICOAGULANTS BERLEX LAB (US) 2002-04-03 EP disclosed
US-5849759-A Naphthyl-substituted benzimidazole derivatives as anti-coagulants BERLEX LABORATORIES, INC. (US) 1998-12-15 US disclosed