SCHEMBL7478093

SCHEMBL7478093

COc1ccc(CC(=O)N2CCC(N3C(=O)OCc4ccccc43)CC2)c(OC)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
OXTR P30559 20/20 1.00
AVPR2 P30518 2/20 0.66
AVPR1A P37288 2/20 0.66
ALDH1A1 P00352 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7441283 0.90 OXTR (0.84) OXTRAVPR2AVPR1AALDH1A1
Hydrochloric Acid SCHEMBL7475350 0.89 OXTR (0.83) OXTRAVPR2AVPR1AALDH1A1
SCHEMBL7357703 0.87 OXTR (0.82) OXTRAVPR2AVPR1AALDH1A1
SCHEMBL7452945 0.85 OXTR (0.79) OXTRAVPR2AVPR1AALDH1A1
SCHEMBL7445878 0.83 OXTR (0.76) OXTRAVPR2AVPR1AALDH1A1
SCHEMBL7439675 0.83 OXTR (0.76) OXTRAVPR2AVPR1AALDH1A1
SCHEMBL7394297 0.82 OXTR (0.79) OXTRAVPR2AVPR1AALDH1A1
SCHEMBL7481810 0.82 OXTR (0.74) OXTRAVPR2AVPR1AALDH1A1
SCHEMBL8093072 0.81 OXTR (0.78) OXTRAVPR2AVPR1AALDH1A1
SCHEMBL8092959 0.81 OXTR (1.00) OXTRAVPR2AVPR1AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0714299-B1 BENZOXAZINONE AND BENZOPYRIMIDINONE PIPERIDINYL TOCOLYTIC OXYTOCIN RECEPTOR ANTAGONISTS MERCK & CO INC (US) 2002-04-24 EP disclosed
US-5665719-A Benzoxazinone and benzopyrimidinone piperidinyl tocolytic oxytocin receptor antagonists MERCK & CO., INC. (US) 1997-09-09 US disclosed