SCHEMBL7478499

SCHEMBL7478499

Nc1[nH]nc(-c2ccccc2F)c1C(=O)c1cccc(OCCN2CCOCC2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 2/20 0.54
KDM4E B2RXH2 1/20 0.46
TP53 P04637 1/20 0.46
TSHR P16473 1/20 0.46
NR1H4 Q96RI1 1/20 0.45
ABCB1 P08183 1/20 0.43
PDGFRB P09619 1/20 0.43
PDGFRA P16234 1/20 0.43
WNT1 P04628 1/20 0.42
DYRK1A Q13627 1/20 0.42
HDAC1 Q13547 1/20 0.42
EPHX2 P34913 4/20 0.42
KEAP1 Q14145 2/20 0.42
NFE2L2 Q16236 2/20 0.42
LCK P06239 1/20 0.42
ADORA3 P0DMS8 1/20 0.42
ADORA2A P29274 1/20 0.42
ADORA2B P29275 1/20 0.42
ADORA1 P30542 1/20 0.42
CNR1 P21554 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5321309 0.87 MAPK14 (0.61) MAPK14KDM4ETP53TSHRNR1H4
Hydrochloric Acid SCHEMBL7466695 0.86 MAPK14 (0.60) MAPK14KDM4ETP53TSHRNR1H4
SCHEMBL7478558 0.84 KDM4E (0.52) MAPK14KDM4ETP53TSHRNR1H4
SCHEMBL5323843 0.76 MAPK14 (0.56) MAPK14WNT1DYRK1AEPHX2
SCHEMBL6163027 0.75 MAPK14 (0.77) MAPK14KDM4ETP53TSHRABCB1
SCHEMBL7475939 0.74 FKBP1A (0.53) MAPK14KDM4EROCK2
SCHEMBL10480077 0.73 KDM4E (0.65) MAPK14KDM4ETP53TSHREPHX2
Hydrochloric Acid SCHEMBL7812345 0.72 MAPK14 (0.62) MAPK14KDM4ETP53TSHREPHX2
SCHEMBL4698008 0.72 KDM4E (0.70) MAPK14KDM4ETP53TSHREPHX2
SCHEMBL4376838 0.71 KDM4E (0.68) MAPK14KDM4ETP53TSHREPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1218346-A1 PYRAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-07-03 EP disclosed
WO-2001021591-A1 PYRAZOLE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2001-03-29 WO disclosed