SCHEMBL7478516

SCHEMBL7478516

CC(C)(C)ON(C=O)c1nc2c([N+](=O)[O-])cccc2[nH]1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKN1 Q16512 1/20 0.44
PKN2 Q16513 1/20 0.44
ADORA3 P0DMS8 1/20 0.41
MGAM O43451 1/20 0.40
GAA P10253 1/20 0.40
SI P14410 1/20 0.40
MGAM2 Q2M2H8 1/20 0.40
PDE10A Q9Y233 1/20 0.35
MEN1 O00255 6/20 0.34
KMT2A Q03164 6/20 0.34
NOS1 P29475 4/20 0.34
NOS2 P35228 3/20 0.33
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 2/20 0.33
CYP1A2 P05177 2/20 0.33
CYP3A4 P08684 2/20 0.33
MAPT P10636 2/20 0.33
TSHR P16473 2/20 0.33
CYP2C19 P33261 2/20 0.33
BLM P54132 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7479831 0.81 MEN1 (0.42) GAAMEN1KMT2AMAPTTDP1
SCHEMBL7966716 0.77 PKN1 (0.55) PKN1PKN2ADORA3MGAMGAA
SCHEMBL7478049 0.71 PKN1 (0.48) PKN1PKN2ADORA3MGAMGAA
SCHEMBL1013588 0.71 PKN1 (0.60) PKN1PKN2ADORA3MGAMGAA
SCHEMBL1548768 0.70 ALDH1A1 (0.43) GAAPDE10AMEN1KMT2AALDH1A1
SCHEMBL8599658 0.70 PKN1 (0.56) PKN1PKN2ADORA3MGAMGAA
SCHEMBL7475814 0.70 PKN1 (0.47) PKN1PKN2ADORA3MGAMGAA
SCHEMBL18776090 0.70 PKN1 (0.52) PKN1PKN2ADORA3MGAMGAA
SCHEMBL6332531 0.69 PKN1 (0.61) PKN1PKN2ADORA3MGAMGAA
SCHEMBL7475180 0.69 PKN1 (0.51) PKN1PKN2ADORA3MGAMGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946519-A1 BENZAMIDE DERIVATIVES HAVING A VASOPRESSIN ANTAGONISTIC ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1999-10-06 EP disclosed
WO-1998024771-A1 BENZAMIDE DERIVATIVES HAVING A VASOPRESSIN ANTAGONISTIC ACTIVITY FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-06-11 WO disclosed