SCHEMBL7478682

SCHEMBL7478682

CCCCc1ccc(NC(=O)Nc2ccc(Oc3ccnc4cc(OC)c(OC)cc34)cc2)cc1

nearest known ligand 0.76

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PDGFRA P16234 18/20 0.76
KDR P35968 18/20 0.76
MET P08581 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7482045 0.92 PDGFRA (0.73) PDGFRAKDR
SCHEMBL5825070 0.92 PDGFRA (0.74) PDGFRAKDRMET
SCHEMBL7482058 0.92 AXL (0.65) PDGFRAKDRMET
SCHEMBL7480693 0.90 PDGFRA (0.82) PDGFRAKDR
SCHEMBL4464828 0.89 FGFR2 (0.73) PDGFRAKDR
SCHEMBL27081475 0.89 PDGFRA (0.95) PDGFRAKDR
SCHEMBL29973354 0.89 PDGFRA (0.95) PDGFRAKDR
SCHEMBL7485360 0.87 PDGFRA (0.75) PDGFRAKDR
SCHEMBL3936662 0.87 KDR (0.74) PDGFRAKDR
SCHEMBL7480326 0.87 FGFR2 (0.67) PDGFRAKDRMET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0860433-B1 QUINOLINE DERIVATIVES AND QUINAZOLINE DERIVATIVES INHIBITING AUTOPHOSPHORYLATION OF GROWTH FACTOR RECEPTOR ORIGINATING IN PLATELET AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KIRIN BREWERY (JP) 2002-07-03 EP claimed
US-6143764-A ETHER DERIVATIVES OF QUINOLINE, ANTITUMOR AGENTS KIRIN BEER KABUSHIKI KAISHA (JP) 2000-11-07 US claimed
EP-0860433-B1 QUINOLINE DERIVATIVES AND QUINAZOLINE DERIVATIVES INHIBITING AUTOPHOSPHORYLATION OF GROWTH FACTOR RECEPTOR ORIGINATING IN PLATELET AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KIRIN BREWERY (JP) 2002-07-03 EP disclosed
US-6143764-A ETHER DERIVATIVES OF QUINOLINE, ANTITUMOR AGENTS KIRIN BEER KABUSHIKI KAISHA (JP) 2000-11-07 US disclosed