SCHEMBL7480326

SCHEMBL7480326

CCCCc1ccc(C(=O)c2ccc(Oc3ccnc4cc(OC)c(OC)cc34)cc2)cc1

nearest known ligand 0.67

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FGFR2 P21802 3/20 0.67
PDGFRA P16234 6/20 0.55
KDR P35968 5/20 0.55
SRC P12931 2/20 0.55
TGFBR1 P36897 2/20 0.55
PDGFRB P09619 2/20 0.54
FLT3 P36888 2/20 0.54
CSF1R P07333 1/20 0.54
FLT4 P35916 1/20 0.54
AURKB Q96GD4 1/20 0.52
MET P08581 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7482058 0.88 AXL (0.65) PDGFRAKDRSRCPDGFRBFLT3
SCHEMBL7478682 0.87 PDGFRA (0.76) PDGFRAKDRMET
SCHEMBL5825897 0.86 PDGFRA (0.52) FGFR2PDGFRAKDRPDGFRBFLT3
SCHEMBL8555453 0.85 PDGFRA (0.52) FGFR2PDGFRAKDRPDGFRBFLT3
SCHEMBL4464828 0.85 FGFR2 (0.73) FGFR2PDGFRAKDRPDGFRBFLT3
SCHEMBL5825070 0.84 PDGFRA (0.74) PDGFRAKDRSRCPDGFRBFLT3
SCHEMBL7481918 0.83 FGFR2 (0.77) FGFR2PDGFRAKDRSRCTGFBR1
SCHEMBL7487378 0.83 FGFR2 (0.77) FGFR2PDGFRAKDRSRCTGFBR1
SCHEMBL7482801 0.82 FGFR2 (0.76) FGFR2PDGFRAKDRSRCTGFBR1
SCHEMBL8069147 0.82 FGFR2 (0.76) FGFR2PDGFRAKDRSRCTGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0860433-B1 QUINOLINE DERIVATIVES AND QUINAZOLINE DERIVATIVES INHIBITING AUTOPHOSPHORYLATION OF GROWTH FACTOR RECEPTOR ORIGINATING IN PLATELET AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KIRIN BREWERY (JP) 2002-07-03 EP claimed
US-6143764-A ETHER DERIVATIVES OF QUINOLINE, ANTITUMOR AGENTS KIRIN BEER KABUSHIKI KAISHA (JP) 2000-11-07 US claimed
EP-0860433-A1 QUINOLINE DERIVATIVES AND QUINAZOLINE DERIVATIVES INHIBITING AUTOPHOSPHORYLATION OF GROWTH FACTOR RECEPTOR ORIGINATING IN PLATELET AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KIRIN BEER KABUSHIKI KAISHA (JP) 1998-08-26 EP claimed
EP-0860433-B1 QUINOLINE DERIVATIVES AND QUINAZOLINE DERIVATIVES INHIBITING AUTOPHOSPHORYLATION OF GROWTH FACTOR RECEPTOR ORIGINATING IN PLATELET AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KIRIN BREWERY (JP) 2002-07-03 EP disclosed
US-6143764-A ETHER DERIVATIVES OF QUINOLINE, ANTITUMOR AGENTS KIRIN BEER KABUSHIKI KAISHA (JP) 2000-11-07 US disclosed
EP-0860433-A1 QUINOLINE DERIVATIVES AND QUINAZOLINE DERIVATIVES INHIBITING AUTOPHOSPHORYLATION OF GROWTH FACTOR RECEPTOR ORIGINATING IN PLATELET AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KIRIN BEER KABUSHIKI KAISHA (JP) 1998-08-26 EP disclosed