SCHEMBL7478908

SCHEMBL7478908

[CH2]CNC(=O)c1ccc(NC(C)=O)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.59
NFKB1 P19838 1/20 0.59
KCNH2 Q12809 1/20 0.59
CACNA1B Q00975 1/20 0.59
APBA1 Q02410 1/20 0.59
SMN1; SMN2 Q16637 4/20 0.57
POLB P06746 2/20 0.57
CYP3A4 P08684 2/20 0.57
NR1H4 Q96RI1 2/20 0.57
THRB P10828 1/20 0.57
BLM P54132 1/20 0.57
ATM Q13315 1/20 0.57
EPHX2 P34913 1/20 0.57
HTT P42858 3/20 0.56
TP53 P04637 1/20 0.54
HIF1A Q16665 1/20 0.54
L3MBTL1 Q9Y468 2/20 0.52
MEN1 O00255 4/20 0.50
KMT2A Q03164 4/20 0.50
HPGD P15428 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12368426 0.84 ALDH1A1 (0.65) ALDH1A1NFKB1KCNH2CACNA1BAPBA1
SCHEMBL13922754 0.82 ALDH1A1 (0.59) ALDH1A1NFKB1KCNH2CACNA1BAPBA1
SCHEMBL11352597 0.82 ALDH1A1 (0.59) ALDH1A1NFKB1KCNH2CACNA1BAPBA1
SCHEMBL6941062 0.81 CACNA1B (0.62) ALDH1A1NFKB1KCNH2CACNA1BAPBA1
SCHEMBL5508324 0.81 ALDH1A1 (0.70) ALDH1A1NFKB1KCNH2CACNA1BAPBA1
SCHEMBL13210697 0.81 CACNA1B (0.85) ALDH1A1CACNA1BAPBA1SMN1; SMN2POLB
SCHEMBL2924725 0.79 CACNA1B (0.65) ALDH1A1NFKB1KCNH2CACNA1BAPBA1
SCHEMBL10755434 0.79 SMN1; SMN2 (0.63) ALDH1A1NFKB1KCNH2CACNA1BAPBA1
SCHEMBL5507897 0.79 SMN1; SMN2 (0.61) ALDH1A1NFKB1KCNH2CACNA1BAPBA1
SCHEMBL11196763 0.79 ALDH1A1 (0.64) ALDH1A1NFKB1KCNH2CACNA1BAPBA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0092830-A2 Cephalosporin derivatives, process for their preparation, pharmaceutical compositions containing them and their application CIBA-GEIGY AG (CH) 1983-11-02 EP claimed
EP-0742903-B1 PIPERIDINE ANALOGS AND CONJUGATES OF PROCAINAMIDE AND NAPA ROCHE DIAGNOSTICS CORP (US) 2002-01-16 EP disclosed
EP-0742903-A4 PIPERIDINE ANALOGS AND CONJUGATES OF PROCAINAMIDE AND NAPA ROCHE DIAGNOSTICS CORP (US) 2000-04-05 EP disclosed
EP-0742903-A1 PIPERIDINE ANALOGS AND CONJUGATES OF PROCAINAMIDE AND NAPA BOEHRINGER MANNHEIM CORPORATION (US) 1996-11-20 EP disclosed
US-5525474-A IMMUNOASSAY; LINKING THE HAPTENIC DRUG VIA ITS MALEIMIDE MOIETY AND A SULFHYDRYL BRIDGE TO AN IMMUNOGENIC CARRIER TO STIMULATE ANTIBODIES BOEHRINGER MANNHEIM CORPORATION (US) 1996-06-11 US disclosed
WO-1995020763-A1 PIPERIDINE ANALOGS AND CONJUGATES OF PROCAINAMIDE AND NAPA BOEHRINGER MANNHEIM CORPORATION (US) 1995-08-03 WO disclosed
EP-0092830-A2 Cephalosporin derivatives, process for their preparation, pharmaceutical compositions containing them and their application CIBA-GEIGY AG (CH) 1983-11-02 EP disclosed