SCHEMBL7478985

SCHEMBL7478985

COc1cc2nccc(Oc3cccc(N)c3)c2cc1OC

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.72
PDGFRB P09619 1/20 0.68
PDGFRA P16234 1/20 0.68
KDR P35968 2/20 0.59
AURKA O14965 1/20 0.58
ABL1 P00519 1/20 0.58
LCK P06239 1/20 0.58
LYN P07948 1/20 0.58
MET P08581 1/20 0.58
TEK Q02763 1/20 0.58
AURKB Q96GD4 1/20 0.58
FGFR2 P21802 2/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7481076 0.87 EGFR (0.78) EGFRPDGFRBPDGFRAFGFR2
SCHEMBL2747998 0.85 PDGFRB (0.71) EGFRPDGFRBPDGFRAKDRAURKA
SCHEMBL19373176 0.85 EGFR (0.74) EGFRPDGFRBPDGFRAKDRFGFR2
SCHEMBL31061546 0.85 EGFR (0.74) EGFRPDGFRBPDGFRAKDRFGFR2
SCHEMBL167396 0.85 PDGFRA (0.74) EGFRPDGFRBPDGFRAKDRFGFR2
SCHEMBL17117826 0.84 FGFR2 (0.78) EGFRPDGFRBPDGFRAKDRFGFR2
SCHEMBL31060325 0.84 FGFR2 (0.78) EGFRPDGFRBPDGFRAKDRFGFR2
SCHEMBL7490337 0.84 EGFR (0.72) EGFRPDGFRBPDGFRAKDRFGFR2
SCHEMBL31060866 0.84 EGFR (0.72) EGFRPDGFRBPDGFRAKDRFGFR2
SCHEMBL31060617 0.84 EGFR (1.00) EGFRPDGFRBPDGFRAKDRFGFR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4662319-A2 PERSONALIZED CRISPR PROFILING FOR CANCER Integrate Bioscience LLC (US) 2025-12-17 EP disclosed
WO-2024168301-A2 PERSONALIZED CRISPR PROFILING FOR CANCER FUNCTION ONCOLOGY, INC. (US) 2024-08-15 WO disclosed
WO-2017049462-A1 NOVEL FLT3 KINASE INHIBITOR AND USES THEREOF 合肥中科普瑞昇生物医药科技有限公司 2017-03-30 WO disclosed
EP-0860433-B1 QUINOLINE DERIVATIVES AND QUINAZOLINE DERIVATIVES INHIBITING AUTOPHOSPHORYLATION OF GROWTH FACTOR RECEPTOR ORIGINATING IN PLATELET AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KIRIN BREWERY (JP) 2002-07-03 EP disclosed
US-6143764-A ETHER DERIVATIVES OF QUINOLINE, ANTITUMOR AGENTS KIRIN BEER KABUSHIKI KAISHA (JP) 2000-11-07 US disclosed
EP-0860433-A1 QUINOLINE DERIVATIVES AND QUINAZOLINE DERIVATIVES INHIBITING AUTOPHOSPHORYLATION OF GROWTH FACTOR RECEPTOR ORIGINATING IN PLATELET AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME KIRIN BEER KABUSHIKI KAISHA (JP) 1998-08-26 EP disclosed