SCHEMBL7479705

SCHEMBL7479705

NCc1nc(-c2nc3c(OC(=O)O)cccc3[nH]2)cs1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 9/20 0.40
CBFB Q13951 2/20 0.39
TP53 P04637 2/20 0.38
ALOX15 P16050 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
HPGD P15428 1/20 0.38
CYP2C19 P33261 1/20 0.38
HSD17B10 Q99714 1/20 0.38
HPSE Q9Y251 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
FKBP1A P62942 1/20 0.36
DHODH Q02127 5/20 0.36
CHEK2 O96017 2/20 0.36
PLK4 O00444 1/20 0.36
MAPK13 O15264 1/20 0.36
DYRK3 O43781 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6587307 0.90 PARP1 (0.42) PARP1CBFBTP53ALOX15SMN1; SMN2
SCHEMBL3159962 0.81 PARP1 (0.61) PARP1DHODHCHEK2PLK4MAPK13
Hydrochloric Acid SCHEMBL6802006 0.80 PARP1 (0.60) PARP1DHODHCHEK2PLK4MAPK13
SCHEMBL7467934 0.74 PARP1 (0.44) PARP1HPSEDHODHCHEK2PLK4
SCHEMBL5879554 0.72 SMN1; SMN2 (0.68) TP53ALOX15SMN1; SMN2ALDH1A1CYP3A4
SCHEMBL3159681 0.70 PARP1 (0.56) PARP1DHODHCHEK2PLK4MAPK13
SCHEMBL6384512 0.68 PARP1 (0.56) PARP1ALOX15HPSEDHODHCHEK2
SCHEMBL7853256 0.67 PARP1 (0.65) PARP1ALOX15HPSEDHODHPKN1
SCHEMBL6590890 0.67 METAP2 (0.50) PARP1CBFBTP53ALOX15SMN1; SMN2
SCHEMBL4975273 0.67 PARP1 (0.40) PARP1TP53ALOX15SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177178-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2002-02-06 EP disclosed
WO-2001082877-A2 USE OF PARP INHIBITORS IN COSMETIC PREPARATIONS BASF AKTIENGESELLSCHAFT (DE) 2001-11-08 WO disclosed
WO-2000068206-A1 HETEROCYCLICALLY SUBSTITUTED BENZIMIDAZOLES, THE PRODUCTION AND APPLICATION THEREOF BASF AKTIENGESELLSCHAFT (DE) 2000-11-16 WO disclosed