SCHEMBL7480294

SCHEMBL7480294

O=CN(Cc1ccccc1)CN1CCN(CCCc2c[nH]c3ccc(-n4cnnc4)cc23)CC1

nearest known ligand 0.74

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 20/20 0.74
HTR1B P28222 20/20 0.74
HTR2A P28223 1/20 0.62
HTR2C P28335 1/20 0.62
HTR1F P30939 1/20 0.62

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7479048 0.85 HTR1D (1.00) HTR1DHTR1BHTR2AHTR2CHTR1F
SCHEMBL7474143 0.84 HTR1D (1.00) HTR1DHTR1B
SCHEMBL7479541 0.81 HTR1D (0.94) HTR1DHTR1B
SCHEMBL7480299 0.80 HTR1D (0.68) HTR1DHTR1B
SCHEMBL7472588 0.79 HTR1D (0.73) HTR1DHTR1B
SCHEMBL7476048 0.79 HTR1D (0.70) HTR1DHTR1B
SCHEMBL7474899 0.79 HTR1D (0.88) HTR1DHTR1BHTR2AHTR2CHTR1F
SCHEMBL8984359 0.79 HTR1D (1.00) HTR1DHTR1B
SCHEMBL4352154 0.78 HTR1D (1.00) HTR1DHTR1B
SCHEMBL8662335 0.78 HTR1D (0.74) HTR1DHTR1BHTR2AHTR2CHTR1F

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0925302-B1 PALLADIUM CATALYZED INDOLIZATION MERCK & CO INC (US) 2002-11-20 EP claimed
EP-0925302-B1 PALLADIUM CATALYZED INDOLIZATION MERCK & CO INC (US) 2002-11-20 EP disclosed
US-5807857-A Piperazine, piperidine and tetrahydropyridine derivative of indol-3-alkyl as 5-HT1D-α agonists MERCK SHARP & DOHME LTD. (GB) 1998-09-15 US disclosed