SCHEMBL7480846

SCHEMBL7480846

Cc1oc(-c2ccccc2)nc1CC=Cc1ccc(CCCC2NC(=O)OC2=O)cc1

nearest known ligand 0.50

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
PPARG P37231 18/20 0.50
PPARA Q07869 14/20 0.50
FFAR1 O14842 1/20 0.39
KDM4E B2RXH2 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8840370 0.95 PPARG (0.51) PPARGPPARAFFAR1KDM4E
SCHEMBL7489094 0.89 PPARG (0.53) PPARGPPARAFFAR1KDM4E
SCHEMBL7487426 0.88 PPARG (0.48) PPARGPPARAFFAR1KDM4E
SCHEMBL7489779 0.88 PPARG (0.53) PPARGPPARAFFAR1
SCHEMBL7488896 0.84 PPARG (0.48) PPARGPPARA
SCHEMBL8794374 0.83 FFAR1 (0.60) PPARGPPARAFFAR1
SCHEMBL7480833 0.82 PPARG (0.50) PPARGPPARAFFAR1KDM4E
SCHEMBL7480829 0.82 PPARG (0.50) PPARGPPARAFFAR1KDM4E
SCHEMBL7486826 0.81 PPARG (0.47) PPARGPPARAFFAR1KDM4E
SCHEMBL7486254 0.81 PPARG (0.49) PPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0643050-B1 Oxazolidinedione derivatives and their use as hypoglycemic agent TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-04-10 EP claimed
EP-0643050-A1 Oxazolidinedione derivatives and their use as hypoglycemic agent Takeda Chemical Industries, Ltd. (JP) 1995-03-15 EP claimed
EP-0643050-B1 Oxazolidinedione derivatives and their use as hypoglycemic agent TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-04-10 EP disclosed
EP-0643050-A1 Oxazolidinedione derivatives and their use as hypoglycemic agent Takeda Chemical Industries, Ltd. (JP) 1995-03-15 EP disclosed