SCHEMBL7489094

SCHEMBL7489094

Cc1oc(-c2ccccc2)nc1CC=Cc1ccc(CC2NC(=O)OC2=O)cc1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PPARG P37231 14/20 0.53
PPARA Q07869 13/20 0.53
KDM4E B2RXH2 1/20 0.41
FFAR1 O14842 1/20 0.37
CYP2C9 P11712 3/20 0.37
CYP3A4 P08684 2/20 0.37
KCNH2 Q12809 2/20 0.37
HPGD P15428 1/20 0.37
MEN1 O00255 1/20 0.36
NPC1 O15118 1/20 0.36
GALR3 O60755 1/20 0.36
MAPT P10636 1/20 0.36
MAPK1 P28482 1/20 0.36
STAT3 P40763 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
HRH3 Q9Y5N1 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8840370 0.91 PPARG (0.51) PPARGPPARAKDM4EFFAR1HRH3
SCHEMBL7480846 0.89 PPARG (0.50) PPARGPPARAKDM4EFFAR1
SCHEMBL7486435 0.83 PPARG (0.53) PPARGPPARAKDM4EFFAR1CYP2C9
SCHEMBL7486432 0.83 PPARG (0.53) PPARGPPARAKDM4EFFAR1CYP2C9
SCHEMBL7909696 0.80 PPARG (0.60) PPARGPPARACYP2C9CYP3A4KCNH2
SCHEMBL7488974 0.79 PPARG (0.45) PPARGPPARAKDM4ECYP2C9CYP3A4
SCHEMBL9721160 0.78 PPARG (0.54) PPARGPPARAKDM4EFFAR1CYP2C9
SCHEMBL9721163 0.78 PPARG (0.54) PPARGPPARAKDM4EFFAR1CYP2C9
SCHEMBL8840367 0.77 PPARG (0.51) PPARGPPARAKDM4EFFAR1
SCHEMBL8840366 0.77 PPARG (0.51) PPARGPPARAKDM4EFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0643050-B1 Oxazolidinedione derivatives and their use as hypoglycemic agent TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-04-10 EP claimed
US-5614544-A HYPOGLYCEMIC AND HYPOLIPIDEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-03-25 US claimed
EP-0643050-A1 Oxazolidinedione derivatives and their use as hypoglycemic agent Takeda Chemical Industries, Ltd. (JP) 1995-03-15 EP claimed
US-5614544-A HYPOGLYCEMIC AND HYPOLIPIDEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-03-25 US disclosed
EP-0643050-A1 Oxazolidinedione derivatives and their use as hypoglycemic agent Takeda Chemical Industries, Ltd. (JP) 1995-03-15 EP disclosed