SCHEMBL7481531

SCHEMBL7481531

[CH2]C(C)Cc1ccc(I)cc1

nearest known ligand 0.61

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.55
CYP2D6 P10635 1/20 0.55
APEX1 P27695 1/20 0.53
PMP22 Q01453 1/20 0.53
SIGMAR1 Q99720 2/20 0.42
CYP3A4 P08684 2/20 0.38
IDO1 P14902 2/20 0.38
APP P05067 2/20 0.37
TAAR1 Q96RJ0 2/20 0.35
SLC6A2 P23975 2/20 0.35
SLC6A3 Q01959 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL662503 0.80 CYP1A2 (0.59) CYP1A2CYP2D6APEX1PMP22SIGMAR1
SCHEMBL10918313 0.78 IDO1 (0.44) CYP1A2IDO1TAAR1SLC6A2SLC6A3
SCHEMBL10922708 0.76 TRPA1 (0.55) IDO1TAAR1
P-Iodoamphetamine SCHEMBL10432865 0.76 TAAR1 (0.61) CYP1A2CYP2D6SIGMAR1TAAR1SLC6A2
P-Iodoamphetamine SCHEMBL1006211 0.76 TAAR1 (0.61) CYP1A2CYP2D6SIGMAR1TAAR1SLC6A2
P-Iodoamphetamine SCHEMBL166055 0.76 TAAR1 (0.61) CYP1A2CYP2D6SIGMAR1TAAR1SLC6A2
SCHEMBL3037011 0.76 SLC6A2 (0.61) IDO1TAAR1SLC6A2SLC6A3
SCHEMBL2454081 0.76 IDO1 (0.48) PMP22IDO1SLC6A2SLC6A3
SCHEMBL1416816 0.76 CYP1A2 (0.55) CYP1A2CYP2D6APEX1PMP22SIGMAR1
SCHEMBL7489625 0.76 TAAR1 (0.61) CYP1A2CYP3A4TAAR1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1177185-A1 4, 5, 6, 7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.p.A. (IT) 2002-02-06 EP disclosed
WO-2000069846-A1 4,5,6,7-TETRAHYDROINDAZOLE DERIVATIVES AS ANTITUMOR AGENTS PHARMACIA & UPJOHN S.P.A. (IT) 2000-11-23 WO disclosed