SCHEMBL7482811

SCHEMBL7482811

COC(=O)c1[nH]c(C)c(C)c1C(C)=O

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.62
CYP1A2 P05177 3/20 0.52
CYP3A4 P08684 1/20 0.52
BRD4 O60885 1/20 0.49
BRPF1 P55201 1/20 0.49
CREBBP Q92793 1/20 0.49
ALDH1A1 P00352 3/20 0.46
MAPK1 P28482 3/20 0.46
SMN1; SMN2 Q16637 3/20 0.44
MAPT P10636 3/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
KDM4E B2RXH2 2/20 0.44
LMNA P02545 1/20 0.44
RAB9A P51151 4/20 0.43
NPC1 O15118 3/20 0.43
PKM P14618 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2150867 0.81 CYP1A2 (0.68) NPSR1CYP1A2ALDH1A1MAPK1SMN1; SMN2
SCHEMBL14123121 0.81 CYP1A2 (0.68) NPSR1CYP1A2CYP3A4BRD4BRPF1
SCHEMBL12531935 0.79 CYP1A2 (0.64) NPSR1CYP1A2ALDH1A1MAPK1SMN1; SMN2
SCHEMBL2150911 0.78 CYP1A2 (0.57) NPSR1CYP1A2CYP3A4BRD4BRPF1
SCHEMBL7256405 0.76 NPSR1 (0.79) NPSR1ALDH1A1MAPK1SMN1; SMN2MAPT
SCHEMBL11282667 0.76 NPSR1 (0.52) NPSR1CYP1A2ALDH1A1MAPK1SMN1; SMN2
SCHEMBL13488596 0.75 NPSR1 (0.66) NPSR1ALDH1A1SMN1; SMN2MAPTMEN1
SCHEMBL14129601 0.74 NPSR1 (0.50) NPSR1CYP1A2ALDH1A1MAPK1SMN1; SMN2
SCHEMBL16506763 0.74 NPSR1 (0.50) NPSR1CYP1A2ALDH1A1MAPK1SMN1; SMN2
SCHEMBL8145766 0.72 CYP1A2 (0.67) NPSR1CYP1A2CYP3A4BRD4BRPF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0742218-B1 PYRROLOPYRIDAZINE DERIVATIVE SANKYO CO (JP) 2002-12-04 EP disclosed
US-6063782-A Pyrrolopyridazine derivatives SANKYO COMPANY, LIMITED (JP) 2000-05-16 US disclosed
EP-0742218-A1 PYRROLOPYRIDAZINE DERIVATIVE SANKYO COMPANY LIMITED (JP) 1996-11-13 EP disclosed