SCHEMBL7256405

SCHEMBL7256405

COC(=O)c1[nH]c(C)c(C(=O)OC)c1C

nearest known ligand 0.79

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.79
RAB9A P51151 4/20 0.66
NPC1 O15118 3/20 0.66
MAPT P10636 5/20 0.63
ALDH1A1 P00352 5/20 0.63
SMN1; SMN2 Q16637 3/20 0.63
KMT2A Q03164 2/20 0.63
KDM4E B2RXH2 2/20 0.63
MEN1 O00255 1/20 0.63
L3MBTL1 Q9Y468 1/20 0.62
HPGD P15428 1/20 0.61
LMNA P02545 2/20 0.60
TSHR P16473 2/20 0.54
POLB P06746 1/20 0.54
MAPK1 P28482 1/20 0.53
HTT P42858 1/20 0.52
TDP1 Q9NUW8 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7252897 0.87 HPGD (0.83) NPSR1RAB9ANPC1MAPTALDH1A1
SCHEMBL7258078 0.87 HPGD (0.83) NPSR1RAB9ANPC1MAPTALDH1A1
SCHEMBL14236103 0.86 NPSR1 (0.70) NPSR1RAB9ANPC1MAPTALDH1A1
SCHEMBL26125904 0.83 ALDH1A1 (0.68) NPSR1RAB9ANPC1MAPTALDH1A1
SCHEMBL12531935 0.83 CYP1A2 (0.64) NPSR1RAB9ANPC1MAPTALDH1A1
SCHEMBL13488596 0.83 NPSR1 (0.66) NPSR1RAB9ANPC1MAPTALDH1A1
SCHEMBL5819637 0.82 MAPT (0.66) NPSR1RAB9ANPC1MAPTALDH1A1
SCHEMBL5819645 0.82 MAPT (0.66) NPSR1RAB9ANPC1MAPTALDH1A1
SCHEMBL7252775 0.81 KMT2A (0.66) NPSR1RAB9ANPC1MAPTALDH1A1
SCHEMBL17278348 0.81 NPSR1 (0.63) NPSR1RAB9ANPC1MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2003035614-A2 TYROSINE KINASE INHIBITORS MERCK & CO., INC. (US) 2003-05-01 WO disclosed
US-6258959-B1 NITROSATION AN ACETOACETATE; REDUCTION; CYCLIZATION BASF AKTIENGESELLSCHAFT (DE) 2001-07-10 US disclosed
US-6166223-A Process for the preparation of 2,4-dimethylpyrrole BASF AKTIENGESELLSCHAFT (DE) 2000-12-26 US disclosed
EP-1013646-A1 Process for the Synthesis of 2,4-Dimethyl-3,5-bis-alkoxy-carbonyl-pyrrole BASF AKTIENGESELLSCHAFT (DE) 2000-06-28 EP disclosed
EP-1013645-A1 Process for the preparation of 2,4-dimethyl-pyrrole BASF AKTIENGESELLSCHAFT (DE) 2000-06-28 EP disclosed