SCHEMBL7483368

SCHEMBL7483368

Cc1oc(-c2ccccc2)nc1CCC(=O)c1ccc(CCC2NC(=O)OC2=O)cc1

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.46
PPARG P37231 18/20 0.44
PPARA Q07869 17/20 0.44
KDM4E B2RXH2 1/20 0.43
PPARD Q03181 4/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7486826 0.95 PPARG (0.47) FFAR1PPARGPPARAKDM4E
SCHEMBL7164860 0.84 PPARG (0.58) PPARGPPARAPPARD
SCHEMBL7489804 0.84 PPARG (0.43) FFAR1PPARGPPARA
SCHEMBL7494345 0.83 PPARG (0.47) FFAR1PPARGPPARAKDM4E
SCHEMBL7487426 0.83 PPARG (0.48) FFAR1PPARGPPARAKDM4E
SCHEMBL7489779 0.83 PPARG (0.53) FFAR1PPARGPPARA
SCHEMBL7483358 0.82 FFAR1 (0.46) FFAR1PPARGPPARAKDM4EPPARD
SCHEMBL7160623 0.81 FFAR1 (0.62) FFAR1PPARGPPARAPPARD
SCHEMBL7488896 0.81 PPARG (0.48) PPARGPPARAPPARD
SCHEMBL7489196 0.81 FFAR1 (0.50) FFAR1PPARGPPARAKDM4EPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0643050-B1 Oxazolidinedione derivatives and their use as hypoglycemic agent TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-04-10 EP disclosed
US-5614544-A HYPOGLYCEMIC AND HYPOLIPIDEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-03-25 US disclosed
EP-0643050-A1 Oxazolidinedione derivatives and their use as hypoglycemic agent Takeda Chemical Industries, Ltd. (JP) 1995-03-15 EP disclosed