SCHEMBL7483358

SCHEMBL7483358

Cc1oc(-c2ccccc2)nc1CCC(=O)c1ccc(CCC2OC(=O)NC2=O)cc1

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.46
PPARG P37231 18/20 0.46
PPARA Q07869 17/20 0.46
KDM4E B2RXH2 1/20 0.43
PPARD Q03181 5/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7486812 0.95 PPARG (0.48) FFAR1PPARGPPARA
SCHEMBL9097431 0.92 PPARG (0.48) FFAR1PPARGPPARAKDM4EPPARD
SCHEMBL7164855 0.85 PPARG (0.62) PPARGPPARAPPARD
SCHEMBL7489790 0.84 PPARG (0.46) FFAR1PPARGPPARA
SCHEMBL7489783 0.84 PPARG (0.46) FFAR1PPARGPPARA
SCHEMBL7494333 0.83 PPARG (0.47) PPARGPPARA
SCHEMBL7485799 0.83 PPARG (0.53) PPARGPPARA
SCHEMBL7489773 0.83 PPARG (0.53) PPARGPPARA
SCHEMBL7483368 0.82 FFAR1 (0.46) FFAR1PPARGPPARAKDM4EPPARD
SCHEMBL8795234 0.81 FFAR1 (0.62) FFAR1PPARGPPARAPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0643050-B1 Oxazolidinedione derivatives and their use as hypoglycemic agent TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-04-10 EP disclosed
US-5614544-A HYPOGLYCEMIC AND HYPOLIPIDEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-03-25 US disclosed
EP-0643050-A1 Oxazolidinedione derivatives and their use as hypoglycemic agent Takeda Chemical Industries, Ltd. (JP) 1995-03-15 EP disclosed