SCHEMBL7486239

SCHEMBL7486239

Cc1oc(-c2ccc3ccccc3c2)nc1C=Cc1ccc(C(=O)O)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.46
CTRC Q99895 1/20 0.45
SLC16A3 O15427 1/20 0.43
SMN1; SMN2 Q16637 3/20 0.41
ALDH1A1 P00352 2/20 0.41
CYP1A2 P05177 2/20 0.41
HSD17B10 Q99714 2/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2C9 P11712 1/20 0.41
HPGD P15428 1/20 0.41
TSHR P16473 1/20 0.41
CYP1B1 Q16678 1/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
POLB P06746 1/20 0.41
CSNK2A1 P68400 1/20 0.40
UTRN P46939 1/20 0.40
RARA P10276 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7486231 1.00 KDM4E (0.46) KDM4ECTRCSLC16A3SMN1; SMN2ALDH1A1
SCHEMBL7482810 0.88 KDM4E (0.46) KDM4ESMN1; SMN2ALDH1A1CYP1A2HSD17B10
SCHEMBL7482819 0.88 KDM4E (0.46) KDM4ESMN1; SMN2ALDH1A1CYP1A2HSD17B10
SCHEMBL7482815 0.88 KDM4E (0.46) KDM4ESMN1; SMN2ALDH1A1CYP1A2HSD17B10
SCHEMBL7491650 0.88 NPC1 (0.50) KDM4ESMN1; SMN2ALDH1A1HPGDNPC1
SCHEMBL7491664 0.88 NPC1 (0.50) KDM4ESMN1; SMN2ALDH1A1HPGDNPC1
SCHEMBL7486298 0.85 KDM4E (0.46) KDM4ESMN1; SMN2ALDH1A1CYP1A2HSD17B10
SCHEMBL7486296 0.85 KDM4E (0.46) KDM4ESMN1; SMN2ALDH1A1CYP1A2HSD17B10
SCHEMBL7481919 0.83 KDM4E (0.45) KDM4ESMN1; SMN2ALDH1A1CYP1A2HSD17B10
SCHEMBL7481914 0.83 KDM4E (0.45) KDM4ESMN1; SMN2ALDH1A1CYP1A2HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0643050-B1 Oxazolidinedione derivatives and their use as hypoglycemic agent TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2002-04-10 EP disclosed
US-5614544-A HYPOGLYCEMIC AND HYPOLIPIDEMIC AGENTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-03-25 US disclosed
EP-0643050-A1 Oxazolidinedione derivatives and their use as hypoglycemic agent Takeda Chemical Industries, Ltd. (JP) 1995-03-15 EP disclosed