SCHEMBL7487168

SCHEMBL7487168

OCC(OCc1ccccc1)c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.49

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 16/20 0.49
CACNA1F O60840 1/20 0.46
CACNA1D Q01668 1/20 0.46
CACNA1S Q13698 1/20 0.46
CACNA1C Q13936 1/20 0.46
IDO1 P14902 1/20 0.43
TDO2 P48775 1/20 0.43
ACP3 P15309 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7476736 1.00 TACR1 (0.49) TACR1CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL5418286 0.79 CHRNB2 (0.53) TACR1IDO1
SCHEMBL14945152 0.79 CHRNB2 (0.53) TACR1IDO1
SCHEMBL6959276 0.74 TACR1 (0.45) TACR1
SCHEMBL6997883 0.73 TACR1 (0.63) TACR1CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL7000528 0.73 TACR1 (0.63) TACR1CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL6482147 0.73 TACR1 (0.67) TACR1
SCHEMBL6483982 0.73 TACR1 (0.67) TACR1
SCHEMBL6483987 0.73 TACR1 (0.67) TACR1
SCHEMBL6495575 0.73 TACR1 (0.67) TACR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1165540-A1 TETRAHYDROPYRAN DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LTD. (GB) 2002-01-02 EP disclosed
WO-2000056727-A1 TETRAHYDROPYRAN DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME LIMITED (GB) 2000-09-28 WO disclosed