SCHEMBL7487283

SCHEMBL7487283

ClC(Cl)c1ccc2c(c1)OCO2

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.51
CYP1A2 P05177 2/20 0.51
CYP2D6 P10635 2/20 0.51
CYP2C9 P11712 2/20 0.51
CYP2C19 P33261 2/20 0.51
MAPK1 P28482 2/20 0.51
ACHE P22303 3/20 0.47
SMAD3 P84022 1/20 0.46
SLC6A4 P31645 1/20 0.44
P4HB P07237 2/20 0.44
MAPK9 P45984 1/20 0.44
ALDH1A1 P00352 2/20 0.44
HSD17B10 Q99714 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
MAOB P27338 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
ABCG2 Q9UNQ0 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29186227 0.83 CYP3A4 (0.49) CYP3A4CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL10823820 0.83 CYP3A4 (0.51) CYP3A4CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL354059 0.83 SLC6A4 (0.50) CYP3A4CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL108101 0.82 CYP3A4 (0.55) CYP3A4CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL2661346 0.78 SLC6A4 (0.53) CYP3A4CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL11217449 0.78 CYP3A4 (0.54) CYP3A4CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL7898797 0.78 CYP3A4 (0.54) CYP3A4CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL1599758 0.78 CYP3A4 (0.54) CYP3A4CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL108228 0.78 CYP3A4 (0.54) CYP3A4CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL18626121 0.78 CYP3A4 (0.54) CYP3A4CYP1A2CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5696301-A Process for preparing protocatechualdehyde UBE INDUSTRIES, LTD. (JP) 1997-12-09 US claimed
EP-0786446-A1 Process for preparing protocatechualdehyde UBE INDUSTRIES, LTD. (JP) 1997-07-30 EP claimed
JP-9263563-A None JP disclosed
JP-9263562-A None JP disclosed
EP-1242075-A4 INDOLE COMPOUNDS SMITHKLINE BEECHAM CORP (US) 2002-12-04 EP disclosed
EP-1242075-A2 INDOLE COMPOUNDS SmithKline Beecham Corporation (US) 2002-09-25 EP disclosed
CN-1070835-C Method for preparation of protocatechuic aldehyde UBE INDUSTRIES (JP) 2001-09-12 CN disclosed
WO-2001030752-A2 INDOLE COMPOUNDS FOR TREATING BACTERIAL INFECTIONS SMITHKLINE BEECHAM CORPORATION (US) 2001-05-03 WO disclosed
US-5856509-A HYPOTENSIVE AGENTS ROUSSEL UCLAF (FR) 1999-01-05 US disclosed
US-5696301-A Process for preparing protocatechualdehyde UBE INDUSTRIES, LTD. (JP) 1997-12-09 US disclosed
US-5696301-A Process for preparing protocatechualdehyde UBE INDUSTRIES, LTD. (JP) 1997-12-09 US disclosed
EP-0786446-A1 Process for preparing protocatechualdehyde UBE INDUSTRIES, LTD. (JP) 1997-07-30 EP disclosed
EP-0786446-A1 Process for preparing protocatechualdehyde UBE INDUSTRIES, LTD. (JP) 1997-07-30 EP disclosed
US-5126461-A Silica in organic solution SHELL RESEARCH LIMITED (GB) 1992-06-30 US disclosed
EP-0432818-A2 Process for opening cyclopropane rings SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1991-06-19 EP disclosed
US-4849420-A HYPOTENSIVE AGENTS AMERICAN HOME PRODUCTS CORPORATION (US) 1989-07-18 US disclosed
EP-0006978-B1 BENZYL ESTERS WITH FLUORINATED ETHER AND/OR THIOETHER GROUPS, THEIR PREPARATIONS AND THEIR USE AS INSECTICIDES; INTERMEDIATE PRODUCTS AND THEIR PREPARATIONS BAYER AG (DE) 1986-01-29 EP disclosed
EP-0041131-B1 PREPARATION OF FLUORO-SUBSTITUTED BENZODIOXOLES AND BENZODIOXANES BAYER AG (DE) 1984-06-13 EP disclosed
EP-0041131-A2 Preparation of fluoro-substituted benzodioxoles and benzodioxanes BAYER AG (DE) 1981-12-09 EP disclosed
EP-0006978-A2 Benzyl esters with fluorinated ether and/or thioether groups, their preparations and their use as insecticides; intermediate products and their preparations BAYER AG (DE) 1980-01-23 EP disclosed