SCHEMBL7488178

SCHEMBL7488178

CCOC(=O)OC1Nc2cc(Cl)cc(Cl)c2C(c2ccc(OC)cc2)C1c1ccc(OC)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.39
GAA P10253 2/20 0.37
KDM4E B2RXH2 2/20 0.37
HPGD P15428 2/20 0.37
LMNA P02545 1/20 0.37
HSD17B10 Q99714 1/20 0.37
MEN1 O00255 1/20 0.37
TSHR P16473 1/20 0.37
KMT2A Q03164 1/20 0.37
GABRA2 P47869 1/20 0.36
GABRB2 P47870 1/20 0.36
HTT P42858 1/20 0.35
MYLK Q15746 2/20 0.35
ACHE P22303 2/20 0.35
BCHE P06276 1/20 0.35
THRB P10828 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6950793 0.96 ALDH1A1 (0.38) ALDH1A1GAAKDM4EHPGDLMNA
SCHEMBL6766668 0.84 ALDH1A1 (0.44) ALDH1A1GAAKDM4EHPGDLMNA
SCHEMBL6766686 0.81 ALDH1A1 (0.48) ALDH1A1MEN1TSHRKMT2A
SCHEMBL7491517 0.79 GAA (0.40) ALDH1A1GAAKDM4ETSHRHTT
SCHEMBL6951562 0.79 CYP2C9 (0.37) CYP2C9CYP2C19
SCHEMBL6765763 0.78 ALDH1A1 (0.44) ALDH1A1GAAKDM4EHPGDLMNA
SCHEMBL7490930 0.76 ALDH1A1 (0.40) ALDH1A1GAAKDM4EHPGDLMNA
SCHEMBL6952696 0.74 KDM4E (0.33) ALDH1A1GAAKDM4EHPGD
SCHEMBL6213758 0.72 POLB (0.33) KDM4ETSHR
SCHEMBL6217832 0.71 MAPK1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1254118-A2 SUBSTITUTED 1,2,3,4- TETRAHYDROQUINOLINE-2-CARBOXYLIC ACID DERIVATIVES Grünenthal GmbH (DE) 2002-11-06 EP disclosed
WO-2001058875-A2 SUBSTITUTED 1,2,3,4- TETRAHYDROQUINOLINE-2-CARBOXYLIC ACID DERIVATIVES Grünenthal GmbH (DE) 2001-08-16 WO disclosed