SCHEMBL7488198

SCHEMBL7488198

CS(=O)(=O)c1ccc(-c2c(-c3ccccc3C(=O)C(=O)c3ccccc3)ccc(C=S)c2Cl)cc1

nearest known ligand 0.40

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 7/20 0.40
AKR1C2 P52895 1/20 0.36
AKR1C1 Q04828 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7085231 0.85 PTGS2 (0.48) PTGS2
SCHEMBL7091359 0.78 PTGS2 (0.45) PTGS2
SCHEMBL7083940 0.78 PTGS2 (0.45) PTGS2AKR1C2AKR1C1
SCHEMBL7084270 0.76 PTGS2 (0.44) PTGS2
SCHEMBL7493552 0.76 PTGS2 (0.44) PTGS2
SCHEMBL7085149 0.75 PTGS2 (0.40) PTGS2
SCHEMBL7089294 0.74 PTGS2 (0.43) PTGS2
SCHEMBL7087953 0.71 PTGS2 (0.46) PTGS2
SCHEMBL7088115 0.71 SLC6A4 (0.42)
SCHEMBL7087484 0.70 PTGS2 (0.41) PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0772601-B1 4,5-SUBSTITUTED IMIDAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION SEARLE & CO (US) 2002-09-18 EP disclosed
US-6426360-B1 ANTIARTHRITIC AGENTS G D SEARLE & CO. 2002-07-30 US disclosed
EP-1211244-A2 4,5-substitued imidazolyl compounds for the treatment of inflammation G.D. Searle & Co. (US) 2002-06-05 EP disclosed
WO-1996003387-A1 4,5-SUBSTITUTED IMIDAZOLYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1996-02-08 WO disclosed