SCHEMBL748827

SCHEMBL748827

O=C(CNCCc1cccc(Br)c1)c1ccc(Cl)cc1

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 3/20 0.58
HDAC1 Q13547 1/20 0.49
HSP90AA1 P07900 1/20 0.48
TAAR1 Q96RJ0 1/20 0.47
EGFR P00533 1/20 0.46
ERBB2 P04626 1/20 0.46
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
PKM P14618 1/20 0.44
MAPT P10636 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
GPR84 Q9NQS5 1/20 0.42
THRB P10828 1/20 0.41
GSK3B P49841 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2298164 0.83 MAPT (0.58) CNR1HDAC1TAAR1NPC1RAB9A
SCHEMBL1013717 0.81 CNR1 (0.68) CNR1HSP90AA1TAAR1NPC1RAB9A
SCHEMBL15785091 0.79 NPC1 (0.51) HSP90AA1TAAR1NPC1RAB9A
SCHEMBL14431556 0.77 TAAR1 (0.54) CNR1TAAR1NPC1RAB9AGPR84
SCHEMBL2293951 0.77 MGLL (0.55) HDAC1HSP90AA1NPC1RAB9AMAPT
SCHEMBL14431603 0.75 TAAR1 (0.59) CNR1TAAR1EGFRERBB2NPC1
SCHEMBL14432356 0.75 TAAR1 (0.55) CNR1TAAR1NPC1RAB9APKM
SCHEMBL18286143 0.75 TSHR (0.54) CNR1NPC1RAB9APKMMAPT
SCHEMBL1025737 0.72 CA12 (0.50) HDAC1HSP90AA1NPC1RAB9AMAPT
SCHEMBL2290144 0.71 MAPT (0.62) HDAC1NPC1RAB9AMAPTL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2429295-A1 ARYL, HETEROARYL, AND HETEROCYCLE SUBSTITUTED TETRAHYDROISOQUINOLINES AND USE THEREOF Albany Molecular Research, Inc. (US) 2012-03-21 EP disclosed
WO-2010132437-A1 ARYL, HETEROARYL, AND HETEROCYCLE SUBSTITUTED TETRAHYDROISOQUINOLINES AND USE THEREOF ALBANY MOLECULAR RESEARCH, INC. (US) 2010-11-18 WO disclosed