SCHEMBL7488394

SCHEMBL7488394

Cc1ccc(NC(=O)Nc2ccccc2Br)c(O)c1C#N.O=C(Nc1ccccc1Br)Nc1cccc(C(=O)Nc2ccccc2)c1O

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CXCR2 P25025 11/20 0.57
CXCR1 P25024 9/20 0.57
RAB9A P51151 3/20 0.49
NPC1 O15118 2/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
HTT P42858 2/20 0.49
LMNA P02545 1/20 0.49
SMN1; SMN2 Q16637 2/20 0.44
HPGD P15428 1/20 0.41
KDM4E B2RXH2 1/20 0.41
GAA P10253 1/20 0.41
ALDH1A1 P00352 1/20 0.41
ADRB3 P13945 1/20 0.41
TSPO P30536 1/20 0.41
SLC6A3 Q01959 1/20 0.41
ABCG2 Q9UNQ0 1/20 0.40
F2R P25116 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3704458 0.87 CXCR2 (0.73) CXCR2CXCR1RAB9ANPC1MEN1
SCHEMBL3715237 0.85 KMT2A (0.68) CXCR2CXCR1RAB9ANPC1MEN1
SCHEMBL7488390 0.80 CXCR2 (0.53) CXCR2CXCR1RAB9ANPC1MEN1
SCHEMBL24421980 0.80 CXCR1 (0.46) CXCR2CXCR1RAB9ANPC1MEN1
SCHEMBL7492930 0.76 CXCR2 (0.72) CXCR2CXCR1MEN1KMT2AHTT
SCHEMBL7487837 0.73 CXCR2 (1.00) CXCR2CXCR1RAB9ANPC1MEN1
SCHEMBL5594974 0.72 KMT2A (0.61) CXCR2CXCR1RAB9ANPC1MEN1
SCHEMBL5595051 0.71 HTT (0.52) CXCR2CXCR1RAB9ANPC1MEN1
SCHEMBL8052698 0.71 KMT2A (0.69) RAB9ANPC1MEN1KMT2AHTT
SCHEMBL3710377 0.70 CXCR2 (0.75) CXCR2CXCR1RAB9ANPC1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0896531-A4 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2002-10-30 EP disclosed
EP-0896531-A1 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1999-02-17 EP disclosed
WO-1997029743-A1 IL-8 RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-08-21 WO disclosed